SCHEMBL31107663

SCHEMBL31107663

COC(=O)c1cc(OCC2(NC(=O)OC(C)(C)C)CCC2)ccc1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.37
PPIA P62937 2/20 0.37
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
ATR Q13535 1/20 0.35
BTK Q06187 1/20 0.35
THRB P10828 1/20 0.35
MAPT P10636 2/20 0.34
KDM4E B2RXH2 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
HPGD P15428 1/20 0.34
CYP2C19 P33261 1/20 0.34
PDK2 Q15119 1/20 0.34
ALOX5AP P20292 1/20 0.33
CA12 O43570 5/20 0.33
CA1 P00915 5/20 0.33
CA2 P00918 5/20 0.33
CA9 Q16790 5/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31107651 0.90 P2RX7 (0.38) P2RX7PPIANPC1RAB9ABTK
SCHEMBL29135649 0.78 P2RX7 (0.36) P2RX7PPIAATRMAPTKDM4E
SCHEMBL31583140 0.77 ATR (0.42) P2RX7PPIAATR
SCHEMBL25155339 0.76 CA12 (0.56) MAPTHPGDPDK2CA12CA1
SCHEMBL30344719 0.76 CA12 (0.56) MAPTHPGDPDK2CA12CA1
SCHEMBL13162402 0.75 CA12 (0.57) CYP2C19PDK2CA12CA1CA2
SCHEMBL2741679 0.74 P2RX7 (0.40) P2RX7PPIANPC1RAB9AMAPT
SCHEMBL31360270 0.74 PPIA (0.36) PPIAPDK2KIT
SCHEMBL25155384 0.74 PPIA (0.36) PPIAPDK2KIT
SCHEMBL25155900 0.73 MTNR1A (0.43) ATRCA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024215817-A1 NOVEL 5-CYCLOPROYLQUINOLINE DERIVATIVES AS PLPRO INHIBITORS PFIZER INC. (US) 2024-10-17 WO disclosed