SCHEMBL3129443

SCHEMBL3129443

CCS(=O)(=O)c1cccc(CC(N)=O)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.37
HTT P42858 1/20 0.35
JAK1 P23458 1/20 0.35
TYK2 P29597 1/20 0.35
PARP1 P09874 1/20 0.35
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
PDE4B Q07343 1/20 0.34
NPSR1 Q6W5P4 2/20 0.34
MBOAT4 Q96T53 1/20 0.34
ALDH1A1 P00352 1/20 0.33
PSIP1 O75475 2/20 0.33
HRH4 Q9H3N8 1/20 0.33
HSD11B1 P28845 1/20 0.32
GRIN2D O15399 2/20 0.32
GRIN3B O60391 2/20 0.32
GRIN1 Q05586 2/20 0.32
GRIN2A Q12879 2/20 0.32
GRIN2B Q13224 2/20 0.32
GRIN2C Q14957 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3121446 0.85 MBOAT4 (0.45) CNR2HTTPARP1CYP3A4CYP2C19
SCHEMBL16234260 0.79 PSIP1 (0.39) JAK1TYK2PARP1NPSR1MBOAT4
SCHEMBL25216536 0.79 MAOB (0.34) CNR2HTTCYP3A4CYP2C19PDE4B
SCHEMBL3928945 0.77 CNR2 (0.47) CNR2JAK1TYK2PARP1NPSR1
SCHEMBL3466817 0.74 CNR2 (0.37) CNR2JAK1TYK2PARP1NPSR1
SCHEMBL29351319 0.74 P2RX7 (0.49) HTTPARP1NPSR1MBOAT4ALDH1A1
SCHEMBL6510299 0.74 P2RX7 (0.49) HTTPARP1NPSR1MBOAT4ALDH1A1
SCHEMBL3466471 0.74 CNR2 (0.35) CNR2JAK1TYK2PARP1NPSR1
SCHEMBL16232198 0.73 PSIP1 (0.34) CNR2HTTJAK1TYK2NPSR1
SCHEMBL3223183 0.72 CPB2 (0.42) HTTNPSR1HRH4GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010036632-A1 AZAINDAZOLE COMPOUNDS AS CCR1 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-01 WO disclosed