SCHEMBL3129599

SCHEMBL3129599

N#CC1=C(N)OC2=C(C(=O)CC(c3ccccc3)C2)C1c1ccc(Br)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.72
MAPT P10636 4/20 0.72
HTT P42858 2/20 0.72
GAA P10253 1/20 0.60
TSHR P16473 2/20 0.57
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
NPSR1 Q6W5P4 2/20 0.47
RECQL P46063 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
GRIA3 P42263 1/20 0.47
GRIA4 P48058 1/20 0.47
TP53 P04637 1/20 0.45
MET P08581 1/20 0.44
USP2 O75604 1/20 0.42
POLB P06746 2/20 0.41
HSD17B10 Q99714 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL562770 0.86 ALDH1A1 (0.68) ALDH1A1MAPTHTTGAATSHR
SCHEMBL3123679 0.83 ALDH1A1 (0.70) ALDH1A1MAPTHTTGAATSHR
SCHEMBL3119482 0.82 ALDH1A1 (0.71) ALDH1A1MAPTHTTGAATSHR
SCHEMBL4084506 0.81 ALDH1A1 (0.67) ALDH1A1MAPTHTTGAATSHR
SCHEMBL4083094 0.80 GAA (0.66) ALDH1A1MAPTGAATSHRMEN1
SCHEMBL3002780 0.78 GAA (0.78) ALDH1A1MAPTHTTGAATSHR
SCHEMBL3005458 0.77 GAA (0.52) ALDH1A1MAPTHTTGAATSHR
SCHEMBL563216 0.77 ALDH1A1 (1.00) ALDH1A1MAPTHTTGAATSHR
SCHEMBL28669991 0.76 ALDH1A1 (0.79) ALDH1A1MAPTTSHRMEN1KMT2A
SCHEMBL28162015 0.76 GAA (1.00) ALDH1A1MAPTHTTGAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010002483-A1 OPTIONALLY CONDENSED DIHYDRO PYRIDINE, DIHYDROPYRIMIDINE AND DIHYDRO PYRANE DERIVATIVES ACTING AS LATE SODIUM CHANNEL BLOCKERS CV THERAPEUTICS, INC. (US) 2010-01-07 WO disclosed
WO-2009006580-A1 OPTIONALLY CONDENSED DIHYDROPYRIDINE, DIHYDROPYRIMIDINE AND DIHYDROPYRANE DERIVATIVES ACTING AS LATE SODIUM CHANNEL BLOCKERS CV THERAPEUTICS, INC. (US) 2009-01-08 WO disclosed