SCHEMBL3130105

SCHEMBL3130105

CCCCCCCC/C=C\CCCCCCCC(=O)O[C@H](COC(=O)CCCCCCCCCCCCC(C)C)COP(=O)([O-])OCC[N+](C)(C)C

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.79
NR5A2 O00482 1/20 0.79
NR5A1 Q13285 1/20 0.79
ALDH1A1 P00352 1/20 0.71
MAPT P10636 1/20 0.70
RECQL P46063 1/20 0.63
FABP3 P05413 1/20 0.63
ADRA1D P25100 1/20 0.54
PTAFR P25105 1/20 0.54
HTR1D P28221 1/20 0.54
HTR2C P28335 1/20 0.54
ADRA1B P35368 1/20 0.54
DRD3 P35462 1/20 0.54
TMEM97 Q5BJF2 1/20 0.54
PRKCE Q02156 1/20 0.53
PRKCQ Q04759 1/20 0.53
PRKCD Q05655 1/20 0.53
PRKCA P17252 1/20 0.53
SELP P16109 1/20 0.52
ENPP2 Q13822 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18037179 1.00 SMN1; SMN2 (0.79) SMN1; SMN2NR5A2NR5A1ALDH1A1MAPT
SCHEMBL15709161 0.95 SMN1; SMN2 (0.88) SMN1; SMN2NR5A2NR5A1ALDH1A1MAPT
SCHEMBL416515 0.95 SMN1; SMN2 (0.88) SMN1; SMN2NR5A2NR5A1ALDH1A1MAPT
SCHEMBL234634 0.95 SMN1; SMN2 (0.88) SMN1; SMN2NR5A2NR5A1ALDH1A1MAPT
SCHEMBL25354838 0.95 SMN1; SMN2 (0.88) SMN1; SMN2NR5A2NR5A1ALDH1A1MAPT
SCHEMBL23188433 0.95 SMN1; SMN2 (0.88) SMN1; SMN2NR5A2NR5A1ALDH1A1MAPT
SCHEMBL235532 0.95 SMN1; SMN2 (0.88) SMN1; SMN2NR5A2NR5A1ALDH1A1MAPT
SCHEMBL45162 0.95 SMN1; SMN2 (0.88) SMN1; SMN2NR5A2NR5A1ALDH1A1MAPT
SCHEMBL22492184 0.95 SMN1; SMN2 (0.88) SMN1; SMN2NR5A2NR5A1ALDH1A1MAPT
SCHEMBL178155 0.95 SMN1; SMN2 (0.88) SMN1; SMN2NR5A2NR5A1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4729052-A1 SUSTAINED RELEASE DOSAGE FORM FOR LOW SOLUBILITY COMPOUND TETRAHYDROCANNABINOL AND METHODS FOR PREPARING OF THIS SUSTAINED RELEASE DOSAGE FORM Emoviar PharmaCon GmbH (DE) 2026-04-22 EP disclosed
EP-4729049-A1 SUSTAINED RELEASE DOSAGE FORM FOR LOW SOLUBILITY COMPOUND AXITINIB AND METHODS FOR PREPARING OF THIS SUSTAINED RELEASE DOSAGE FORM Emoviar PharmaCon GmbH (DE) 2026-04-22 EP disclosed
US-20250281596-A1 IONIZABLE CATIONIC COMPOUND Seqirus Inc. 2025-09-11 US disclosed
US-20250268839-A1 PROMOTING TRAINED IMMUNITY WITH THERAPEUTIC NANOBIOLOGIC COMPOSITIONS STICHTING RADBOUD UNIVERSITAIR MEDISCH CENTRUM (NL) 2025-08-28 US disclosed
EP-4445898-A1 SUSTAINED RELEASE DOSAGE FORMS COMPRISING COMPLEXES OF LOW SOLUTIBILITY COMPOUNDS, AND METHODS FOR THEIR PREPARATION Emoviar PharmaCon GmbH (DE) 2024-10-16 EP disclosed
EP-4445899-A1 SUSTAINED RELEASE DOSAGE FORMS COMPRISING COMPLEXES OF LOW SOLUTIBILITY COMPOUNDS, AND METHODS FOR THEIR PREPARATION Emoviar PharmaCon GmbH (DE) 2024-10-16 EP disclosed
US-20240261223-A1 MODULAR LIPID COMPOUNDS AND TWO- TO THREE-COMPONENT LIPID NANOPARTICLE COMPOSITIONS SUNVAX MRNA THERAPEUTICS (US) 2024-08-08 US disclosed
EP-4351618-A2 TREM-2/DAP-12 INHIBITORS FOR TREATING LUNG DISEASE AND INJURY AND COMBINATIONS THEREOF Signablk, Inc. (US) 2024-04-17 EP disclosed
WO-2022245553-A2 TREM-2/DAP-12 INHIBITORS FOR TREATING LUNG DISEASE AND INJURY AND COMBINATIONS THEREOF SIGNABLK, INC. (US) 2022-11-24 WO disclosed
US-20210214401-A1 MANUFACTURING METHOD OF NANODISC COMPRISING AN OLFACTORY RECEPTOR PROTEIN AND NANODISC COMPRISING AN OLFACTORY RECEPTOR PROTEIN MANUFACTURED BY THE SAME SEOUL NATIONAL UNIVERSITY R&DB FOUNDATION (KR) 2021-07-15 US disclosed
US-20040213833-A1 certain MMP inhibitory peptides improve the targeting of liposomes to cancer cells and enhance the uptake thereof by such cells CTT CANCER TARGETING TECHNOLOGIES OY (FI) 2004-10-28 US disclosed
EP-1469830-A2 METHOD FOR MAKING HOMOGENEOUS SPRAY-DRIED SOLID AMORPHOUS DRUG DISPERSIONS USING PRESSURE NOZZLES Pfizer Products Inc. (US) 2004-10-27 EP disclosed
EP-1438021-A2 METHODS AND APPARATUS FOR EXTRUSION OF VESICLES AT HIGH PRESSURE Esperion Therapeutics Inc. (US) 2004-07-21 EP disclosed
WO-2003063821-A2 METHOD FOR MAKING HOMOGENEOUS SPRAY-DRIED SOLID AMORPHOUS DRUG DISPERSIONS USING PRESSURE NOZZLES PFIZER PRODUCTS INC. (US) 2003-08-07 WO disclosed
WO-2003026588-A2 METHODS AND APPARATUS FOR EXTRUSION OF VESICLES AT HIGH PRESSURE ESPERION THERAPEUTICS, INC. (US) 2003-04-03 WO disclosed
US-20030017520-A1 High-efficiency assay for protein mannosyl transferases PHARMACIA & UPJOHN COMPANY 2003-01-23 US disclosed
EP-1260591-A1 High-efficiency assay for protein mannosyl transferases Pharmacia & Upjohn Company (US) 2002-11-27 EP disclosed
US-6099857-A LIPID, VESICLE KIT; DRUG DELIVERY WASHINGTON UNIVERSITY (US) 2000-08-08 US disclosed
WO-1997021729-A9 METHODS AND COMPOSITIONS FOR MODULATING VESICLE RELEASE 1997-11-06 WO disclosed
WO-1995031183-A1 CELL MEMBRANE FUSION COMPOSITION AND METHOD WASHINGTON UNIVERSITY (US) 1995-11-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250281596-A1 IONIZABLE CATIONIC COMPOUND SLC11A2, ABCB4, ARG2 SMN1; SMN2 1684/4885NR5A2 2715/4885NR5A1 3268/4885
US-20240261223-A1 MODULAR LIPID COMPOUNDS AND TWO- TO THREE-COMPONENT LIPID NANOPARTICLE COMPOSITIONS PLIN3, PHOSPHO1, SGMS2 SMN1; SMN2 3060/4885NR5A2 4080/4885NR5A1 4504/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.