SCHEMBL3138975

SCHEMBL3138975

CCOC(=O)[C@H](C)n1cccn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 2/20 0.40
MAPT P10636 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KDM4E B2RXH2 6/20 0.36
ALDH1A1 P00352 5/20 0.36
HPGD P15428 4/20 0.36
GLA P06280 1/20 0.36
HSD17B10 Q99714 3/20 0.36
FPR2 P25090 1/20 0.36
PDE4A P27815 1/20 0.35
LMNA P02545 3/20 0.35
TSHR P16473 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
POLB P06746 1/20 0.35
RAB9A P51151 1/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4083681 1.00 NLRP3 (0.40) NLRP3MAPTL3MBTL1KDM4EALDH1A1
SCHEMBL5591669 0.84 NLRP3 (0.41) NLRP3KDM4EALDH1A1HPGDHSD17B10
SCHEMBL30697576 0.82 KMT2A (0.38) NLRP3MAPTKDM4EALDH1A1TSHR
SCHEMBL10362298 0.82 KMT2A (0.38) NLRP3MAPTKDM4EALDH1A1TSHR
SCHEMBL17869461 0.79 MEN1 (0.42) NLRP3KDM4EALDH1A1HPGDHSD17B10
SCHEMBL10513126 0.79 FDPS (0.36) ALDH1A1TSHRMEN1KMT2ACYP1A2
SCHEMBL21672154 0.79 ALDH1A1 (0.46) MAPTL3MBTL1ALDH1A1HPGDHSD17B10
SCHEMBL27710074 0.77 MEN1 (0.35) ALDH1A1TSHRMEN1KMT2AFDPS
SCHEMBL29427328 0.77 MEN1 (0.32) MEN1KMT2A
SCHEMBL24900643 0.76 ALDH1A1 (0.36) NLRP3KDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054427-B1 AVERMECTIN DERIVATIVES BAYER CROPSCIENCE AG (DE) 2010-07-14 EP disclosed
CN-101528761-A Avermectin derivatives BAYER CROPSCIENCE AG (DE) 2009-09-09 CN disclosed
EP-2054427-A2 AVERMECTIN DERIVATIVES Bayer CropScience AG (DE) 2009-05-06 EP disclosed
WO-2008019784-A2 AVERMECTIN DERIVATIVES BAYER CROPSCIENCE AG (DE) 2008-02-21 WO disclosed