SCHEMBL27710074

SCHEMBL27710074

CC(C(=O)C(C)n1cccn1)n1cccn1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ADRB3 P13945 3/20 0.34
NOS1 P29475 2/20 0.33
ELANE P08246 2/20 0.33
ALDH1A1 P00352 1/20 0.32
FDPS P14324 1/20 0.32
MGLL Q99685 1/20 0.31
TSHR P16473 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6434486 0.85 MEN1 (0.37) MEN1KMT2AADRB3NOS1ELANE
SCHEMBL4663219 0.85 ALDH1A1 (0.43) MEN1KMT2AADRB3NOS1ELANE
SCHEMBL3091768 0.85 ALDH1A1 (0.43) MEN1KMT2AADRB3NOS1ELANE
SCHEMBL31354980 0.85 ALDH1A1 (0.43) MEN1KMT2AADRB3NOS1ELANE
SCHEMBL14743754 0.83 NOS1 (0.39) MEN1KMT2AADRB3NOS1ELANE
SCHEMBL10513126 0.80 FDPS (0.36) MEN1KMT2AADRB3NOS1ALDH1A1
SCHEMBL30697576 0.80 KMT2A (0.38) MEN1KMT2AADRB3ALDH1A1TSHR
SCHEMBL10362298 0.80 KMT2A (0.38) MEN1KMT2AADRB3ALDH1A1TSHR
SCHEMBL19292029 0.80 ADRB3 (0.41) MEN1KMT2AADRB3NOS1ELANE
SCHEMBL3138975 0.77 NLRP3 (0.40) MEN1KMT2AALDH1A1FDPSTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105209470-A 6-bridged heteroaryldihydropyrimidines for the treatment and prophylaxis of hepatitis b virus infection HOFFMANN LA ROCHE 2015-12-30 CN disclosed
CN-101212973-B 4-phenyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline derivatives as medicaments for the treatment of infertility ORGANON NV 2011-11-16 CN disclosed
CN-101212973-A 4-phenyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline derivatives as medicaments for the treatment of infertility ORGANON NV (NL) 2008-07-02 CN disclosed