SCHEMBL3142552

SCHEMBL3142552

O=C(O)NCC1(CNc2cnc(Cl)c(-c3cccnc3)c2)CC1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.41
MCHR1 Q99705 4/20 0.40
EGLN3 Q9H6Z9 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
CYP11B2 P19099 1/20 0.36
IDO1 P14902 1/20 0.36
P2RX7 Q99572 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CNR1 P21554 1/20 0.35
KDR P35968 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3143340 0.89 ADORA2B (0.34)
SCHEMBL3146187 0.86 MAP4K4 (0.38) EGLN3P2RX7CNR1
SCHEMBL3151357 0.82 ABL1 (0.42) ABL1MCHR1EGLN3
SCHEMBL3152373 0.82 EGLN1 (0.41) EGLN3P2RX7
SCHEMBL3142555 0.80 ABL1 (0.39) ABL1MCHR1CYP11B2IDO1
SCHEMBL3146697 0.78 ABL1 (0.39) ABL1MCHR1
SCHEMBL3156236 0.78 ALDH1A1 (0.33) CYP11B2KMT2A
Hydrochloric Acid SCHEMBL3775074 0.78 ABL1 (0.38) ABL1MCHR1
SCHEMBL4818188 0.74 KCNQ3 (0.43)
SCHEMBL3147012 0.73 FFAR4 (0.44) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979321-B9 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2010-02-17 EP disclosed
EP-1979321-B1 NOVEL PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINES, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SERVIER LAB (FR) 2009-07-29 EP disclosed