SCHEMBL3147724

SCHEMBL3147724

O=[C]c1nc2ccncc2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
SMN1; SMN2 Q16637 5/20 0.46
PKM P14618 4/20 0.46
KDM4E B2RXH2 4/20 0.46
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
HPGD P15428 2/20 0.46
METAP1 P53582 2/20 0.45
METAP2 P50579 1/20 0.45
HPSE Q9Y251 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
AURKA O14965 1/20 0.43
RPS6KA5 O75582 1/20 0.42
PDE5A O76074 3/20 0.41
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40
NFKB1 P19838 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
KRAS P01116 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9452004 0.85 PDE3B (0.42) ALDH1A1PKMKDM4EMETAP2PDE3B
SCHEMBL14629339 0.81 PSMB8 (0.53) ALDH1A1SMN1; SMN2PKMKDM4ENPC1
SCHEMBL222527 0.75 ALDH1A1 (0.54) ALDH1A1SMN1; SMN2PKMKDM4ENPC1
SCHEMBL1170780 0.74 ALDH1A1 (0.68) ALDH1A1SMN1; SMN2PKMKDM4ENPC1
SCHEMBL34462940 0.71 SMN1; SMN2 (0.50) ALDH1A1SMN1; SMN2PKMKDM4ENPC1
SCHEMBL21496798 0.71 ALDH1A1 (0.50) ALDH1A1SMN1; SMN2PKMKDM4ENPC1
SCHEMBL2106050 0.71 SMN1; SMN2 (0.50) ALDH1A1SMN1; SMN2PKMKDM4ENPC1
SCHEMBL15088513 0.71 SMN1; SMN2 (0.50) ALDH1A1SMN1; SMN2PKMKDM4ENPC1
SCHEMBL9698797 0.71 ALDH1A1 (0.55) ALDH1A1SMN1; SMN2PKMKDM4ENPC1
SCHEMBL7249651 0.71 SMN1; SMN2 (0.50) ALDH1A1SMN1; SMN2PKMKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2233493-A1 Macrolides Pfizer Products Inc. (US) 2010-09-29 EP disclosed
EP-1836211-B1 MACROLIDES PFIZER PROD INC (US) 2010-03-03 EP disclosed