SCHEMBL315428

SCHEMBL315428

Cc1onc(-c2c(Cl)cccc2Cl)c1C(=O)NC1CCC(Cc2ccccc2)(N2CCCC2)CC1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 5/20 0.56
KMT2A Q03164 3/20 0.54
MEN1 O00255 2/20 0.51
ALDH1A1 P00352 3/20 0.50
GAA P10253 2/20 0.50
MAPT P10636 2/20 0.50
KDM4E B2RXH2 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
TSHR P16473 1/20 0.49
PTGS2 P35354 2/20 0.49
ABCB11 O95342 1/20 0.46
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL316302 0.99 GHSR (0.56) GHSRKMT2AMEN1ALDH1A1GAA
SCHEMBL316059 0.95 KMT2A (0.59) GHSRKMT2AMEN1ALDH1A1MAPT
SCHEMBL315461 0.92 KMT2A (0.65) GHSRKMT2AMEN1ALDH1A1GAA
SCHEMBL316051 0.92 KMT2A (0.67) GHSRKMT2AMEN1ALDH1A1GAA
SCHEMBL316159 0.84 KMT2A (0.58) GHSRKMT2AMEN1ALDH1A1GAA
SCHEMBL314979 0.84 GHSR (0.62) GHSRKMT2AMEN1ALDH1A1GAA
SCHEMBL1514721 0.82 KMT2A (0.70) GHSRKMT2AMEN1ALDH1A1GAA
SCHEMBL315998 0.80 KMT2A (0.57) GHSRKMT2AMEN1ALDH1A1GAA
SCHEMBL316299 0.80 KMT2A (0.57) GHSRKMT2AMEN1ALDH1A1MAPT
SCHEMBL316050 0.79 GHSR (0.61) GHSRKMT2AMEN1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US claimed
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US disclosed