SCHEMBL316159

SCHEMBL316159

Cc1onc(-c2c(Cl)cccc2Cl)c1C(=O)NC1CCC(c2ccccc2)(N2CCCCC2)CC1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.58
GHSR Q92847 3/20 0.56
ALDH1A1 P00352 4/20 0.52
GAA P10253 2/20 0.52
MAPT P10636 2/20 0.52
KDM4E B2RXH2 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
PTGS2 P35354 2/20 0.51
TSHR P16473 1/20 0.49
LMNA P02545 1/20 0.47
MEN1 O00255 1/20 0.47
ABCB11 O95342 1/20 0.47
NPSR1 Q6W5P4 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL315998 0.95 KMT2A (0.57) KMT2AGHSRALDH1A1GAAMAPT
SCHEMBL316302 0.85 GHSR (0.56) KMT2AGHSRALDH1A1GAAMAPT
SCHEMBL315428 0.84 GHSR (0.56) KMT2AGHSRALDH1A1GAAMAPT
SCHEMBL315915 0.83 GHSR (0.63) KMT2AGHSRALDH1A1GAAMAPT
Hydrochloric Acid SCHEMBL317007 0.82 GHSR (0.62) KMT2AGHSRALDH1A1GAAMAPT
SCHEMBL316059 0.80 KMT2A (0.59) KMT2AGHSRALDH1A1MAPTKDM4E
SCHEMBL316051 0.78 KMT2A (0.67) KMT2AGHSRALDH1A1GAAMAPT
SCHEMBL1514721 0.78 KMT2A (0.70) KMT2AGHSRALDH1A1GAAMAPT
SCHEMBL315827 0.78 GHSR (0.57) KMT2AGHSRALDH1A1MAPTKDM4E
SCHEMBL315461 0.77 KMT2A (0.65) KMT2AGHSRALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US claimed
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US disclosed