SCHEMBL315857

SCHEMBL315857

Cc1oc(-c2ccc(Cl)cc2)cc1C(=O)NC1CCC(c2cccc(F)c2)(N(C)C)CC1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.43
RAB9A P51151 5/20 0.43
OPRM1 P35372 4/20 0.42
OPRL1 P41146 4/20 0.42
L3MBTL1 Q9Y468 2/20 0.39
MAPK11 Q15759 1/20 0.38
MAPK14 Q16539 1/20 0.38
HPGD P15428 1/20 0.38
ERAP1 Q9NZ08 2/20 0.38
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
ALDH1A1 P00352 1/20 0.37
PKM P14618 1/20 0.37
CNR1 P21554 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL316187 0.79 NPC1 (0.43) NPC1RAB9AL3MBTL1MAPK11MAPK14
SCHEMBL316611 0.76 L3MBTL1 (0.51) NPC1RAB9AOPRM1OPRL1L3MBTL1
SCHEMBL315499 0.75 HSD11B1 (0.42) OPRM1OPRL1KDM4EALDH1A1CNR1
SCHEMBL315547 0.74 GHSR (0.58) L3MBTL1HPGDKDM4ELMNAALDH1A1
Hydrochloric Acid SCHEMBL314995 0.74 GHSR (0.57) HPGDKDM4ELMNAALDH1A1
SCHEMBL316297 0.73 TSHR (0.50) OPRM1OPRL1KDM4ELMNAALDH1A1
SCHEMBL315788 0.73 POLB (0.55) NPC1HPGDLMNAALDH1A1
Hydrochloric Acid SCHEMBL316635 0.73 TSHR (0.49) OPRM1OPRL1KDM4ELMNAALDH1A1
SCHEMBL315615 0.72 KMT2A (0.62) LMNAALDH1A1
SCHEMBL2985751 0.72 CCR3 (0.53) NPC1OPRM1OPRL1KDM4EPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US claimed
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US disclosed