SCHEMBL315499

SCHEMBL315499

CN(C)C1(c2cccc(F)c2)CCC(NC(=O)c2cnn(-c3ccc(Cl)cc3)c2C(F)(F)F)CC1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.42
SPR P35270 1/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CCR1 P32246 2/20 0.40
TRPC3 Q13507 1/20 0.40
OPRL1 P41146 2/20 0.39
NTRK1 P04629 2/20 0.39
OPRM1 P35372 1/20 0.39
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
MAPT P10636 3/20 0.39
GPR6 P46095 1/20 0.39
TP53 P04637 1/20 0.38
CRHR1 P34998 1/20 0.38
HSP90AA1 P07900 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10366974 0.80 HSD11B1 (0.56) HSD11B1SPRKDM4EALDH1A1CCR1
SCHEMBL315879 0.80 CCR1 (0.44) HSD11B1SPRKDM4EALDH1A1CCR1
SCHEMBL316498 0.80 NPSR1 (0.44) HSD11B1SPRKDM4EALDH1A1CCR1
SCHEMBL315779 0.79 HSD11B1 (0.44) HSD11B1SPRKDM4EALDH1A1CCR1
SCHEMBL315976 0.79 KDM4E (0.48) HSD11B1SPRKDM4EALDH1A1CCR1
SCHEMBL2851938 0.79 SPR (0.56) HSD11B1SPRKDM4EALDH1A1TRPC3
SCHEMBL315268 0.78 ALDH1A1 (0.43) HSD11B1SPRKDM4EALDH1A1CCR1
SCHEMBL315723 0.78 ALDH1A1 (0.54) HSD11B1ALDH1A1MAPTTP53
SCHEMBL315441 0.77 KDM4E (0.46) HSD11B1SPRKDM4EALDH1A1CCR1
SCHEMBL316470 0.77 KDM4E (0.43) HSD11B1SPRKDM4EALDH1A1CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US claimed
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US disclosed