SCHEMBL315879

SCHEMBL315879

CN(C)C1(Cc2cccc(Cl)c2)CCC(NC(=O)c2cnn(-c3ccc(Cl)cc3)c2C(F)(F)F)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 3/20 0.44
MAPT P10636 2/20 0.42
HSP90AA1 P07900 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HSD11B1 P28845 1/20 0.41
SPR P35270 1/20 0.41
TRPC3 Q13507 1/20 0.41
TP53 P04637 1/20 0.41
CNR1 P21554 1/20 0.40
CNR2 P34972 1/20 0.40
DRD2 P14416 1/20 0.40
DRD1 P21728 1/20 0.40
GPR6 P46095 1/20 0.40
MGLL Q99685 1/20 0.39
CRHR1 P34998 1/20 0.39
DDR1 Q08345 1/20 0.39
MAPK11 Q15759 1/20 0.39
MAPK14 Q16539 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL315976 0.93 KDM4E (0.48) CCR1MAPTHSP90AA1NPSR1KDM4E
SCHEMBL315779 0.92 HSD11B1 (0.44) CCR1MAPTHSP90AA1NPSR1KDM4E
SCHEMBL315130 0.89 NPC1 (0.45) CCR1MAPTHSP90AA1NPSR1KDM4E
SCHEMBL316498 0.89 NPSR1 (0.44) CCR1MAPTNPSR1KDM4EALDH1A1
SCHEMBL315441 0.86 KDM4E (0.46) CCR1MAPTHSP90AA1NPSR1KDM4E
SCHEMBL316470 0.86 KDM4E (0.43) CCR1MAPTHSP90AA1NPSR1KDM4E
SCHEMBL315268 0.86 ALDH1A1 (0.43) CCR1MAPTNPSR1KDM4EALDH1A1
SCHEMBL315499 0.80 HSD11B1 (0.42) CCR1MAPTHSP90AA1NPSR1KDM4E
SCHEMBL10366974 0.80 HSD11B1 (0.56) CCR1MAPTKDM4EALDH1A1HSD11B1
SCHEMBL10364982 0.79 KDM4E (0.53) MAPTKDM4EALDH1A1HSD11B1SPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US claimed
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US disclosed