SCHEMBL3167014

SCHEMBL3167014

N#Cc1ccc(S(=O)(=O)c2ccc(CO)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.53
CA1 P00915 5/20 0.50
CA2 P00918 5/20 0.50
CA12 O43570 4/20 0.50
CA9 Q16790 3/20 0.50
CA4 P22748 2/20 0.50
CA7 P43166 2/20 0.50
BCHE P06276 1/20 0.50
ACHE P22303 1/20 0.50
CA6 P23280 1/20 0.50
CA5A P35218 1/20 0.50
CA14 Q9ULX7 1/20 0.50
CA5B Q9Y2D0 1/20 0.50
MAPT P10636 1/20 0.49
NAMPT P43490 4/20 0.47
CYP2A6 P11509 1/20 0.44
LOXL2 Q9Y4K0 1/20 0.44
TAS2R14 Q9NYV8 1/20 0.43
TSHR P16473 1/20 0.43
HSD11B1 P28845 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8514633 0.84 CA2 (0.59) CYP19A1CA1CA2CA12CA9
SCHEMBL92970 0.84 LOXL2 (0.58) CYP19A1CA1CA2CA12CA9
SCHEMBL156259 0.84 CA2 (0.67) CA1CA2CA12CA9CA4
SCHEMBL3173425 0.84 CYP19A1 (0.51) CYP19A1CA1CA2CA12CA9
SCHEMBL3174749 0.84 NAMPT (0.52) CYP19A1CA1CA2CA12CA9
SCHEMBL27707919 0.82 LOXL2 (0.56) CYP19A1CA2CA12CA9CA6
Hydrogen Sulfide SCHEMBL27473257 0.82 LOXL2 (0.56) CYP19A1CA2CA12CA9CA6
SCHEMBL27962507 0.80 MAPT (0.59) CYP19A1CA1CA2CA12CA9
SCHEMBL7935644 0.79 CA2 (0.67) CYP19A1CA1CA2CA12CA9
Phosphoric Acid SCHEMBL28852152 0.79 LOXL2 (0.48) CYP19A1CA1CA2CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101061105-B Potentiators of glutamate receptors LILLY CO ELI 2012-05-30 CN disclosed
EP-1817300-B1 POTENTIATORS OF GLUTAMATE RECEPTORS LILLY CO ELI (US) 2010-03-17 EP disclosed
CN-101061105-A Potentiators of glutamate receptors LILLY CO ELI (US) 2007-10-24 CN disclosed