SCHEMBL316737

SCHEMBL316737

CCCc1c(C(=O)NC2CCC(Cc3ccc(F)cc3)(N(C)C)CC2)cnn1-c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.52
POLB P06746 2/20 0.52
MAPK1 P28482 4/20 0.51
MAPK14 Q16539 3/20 0.51
MAPT P10636 6/20 0.47
GAA P10253 2/20 0.46
RAB9A P51151 1/20 0.46
LMNA P02545 2/20 0.43
THRB P10828 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL315859 0.85 MAPT (0.47) ALDH1A1POLBMAPK1MAPK14MAPT
SCHEMBL315723 0.81 ALDH1A1 (0.54) ALDH1A1POLBMAPK1MAPK14MAPT
SCHEMBL316233 0.80 ALDH1A1 (0.49) ALDH1A1POLBMAPK1MAPK14MAPT
SCHEMBL2856262 0.80 ALDH1A1 (0.59) ALDH1A1POLBMAPK1MAPK14MAPT
SCHEMBL316498 0.78 NPSR1 (0.44) ALDH1A1MAPK14MAPT
SCHEMBL2979180 0.76 CCR3 (0.56) ALDH1A1MAPTGAA
SCHEMBL15889273 0.76 POLB (0.58) ALDH1A1POLBMAPK1MAPTGAA
SCHEMBL18016194 0.76 ALDH1A1 (0.52) ALDH1A1POLBMAPK1MAPK14MAPT
SCHEMBL315976 0.75 KDM4E (0.48) ALDH1A1POLBMAPK14MAPT
SCHEMBL316308 0.75 KCNH2 (0.46) POLBMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US claimed
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US disclosed