SCHEMBL315859

SCHEMBL315859

CCCc1c(C(=O)NC2CCC(Cc3ccccc3Cl)(N(C)C)CC2)cnn1-c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.47
GAA P10253 2/20 0.47
ALDH1A1 P00352 8/20 0.46
MAPK1 P28482 4/20 0.46
MAPK14 Q16539 3/20 0.45
POLB P06746 2/20 0.44
LMNA P02545 3/20 0.43
THRB P10828 1/20 0.43
PKM P14618 1/20 0.43
HSD11B1 P28845 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL316737 0.85 ALDH1A1 (0.52) MAPTGAAALDH1A1MAPK1MAPK14
SCHEMBL2856262 0.80 ALDH1A1 (0.59) MAPTGAAALDH1A1MAPK1MAPK14
SCHEMBL316233 0.77 ALDH1A1 (0.49) MAPTGAAALDH1A1MAPK1MAPK14
SCHEMBL315723 0.76 ALDH1A1 (0.54) MAPTGAAALDH1A1MAPK1MAPK14
SCHEMBL15889273 0.76 POLB (0.58) MAPTGAAALDH1A1MAPK1POLB
SCHEMBL2984830 0.75 ALDH1A1 (0.53) MAPTGAAALDH1A1POLB
SCHEMBL316216 0.75 KCNH2 (0.46) MAPTGAAPOLBLMNAPKM
SCHEMBL1403425 0.74 HSD11B1 (0.56) MAPTGAAALDH1A1MAPK1MAPK14
SCHEMBL18016194 0.74 ALDH1A1 (0.52) MAPTGAAALDH1A1MAPK1MAPK14
SCHEMBL14097125 0.74 ALDH1A1 (0.67) MAPTGAAALDH1A1MAPK1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US claimed
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US disclosed