SCHEMBL316233

SCHEMBL316233

CCCc1c(C(=O)NC2CCC(Cc3ccccc3)(N3CCCCCC3)CC2)cnn1-c1ccccc1

nearest known ligand 0.69

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.49
MAPT P10636 5/20 0.49
MAPK1 P28482 4/20 0.48
GAA P10253 2/20 0.48
LMNA P02545 2/20 0.46
THRB P10828 1/20 0.46
POLB P06746 2/20 0.46
MAPK14 Q16539 2/20 0.45
SPR P35270 1/20 0.45
HSD11B1 P28845 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2856262 0.84 ALDH1A1 (0.59) ALDH1A1MAPTMAPK1GAALMNA
SCHEMBL15889273 0.82 POLB (0.58) ALDH1A1MAPTMAPK1GAALMNA
SCHEMBL316737 0.80 ALDH1A1 (0.52) ALDH1A1MAPTMAPK1GAALMNA
SCHEMBL18016194 0.80 ALDH1A1 (0.52) ALDH1A1MAPTMAPK1GAALMNA
SCHEMBL315859 0.77 MAPT (0.47) ALDH1A1MAPTMAPK1GAALMNA
SCHEMBL315633 0.76 KCNH2 (0.44) ALDH1A1MAPTLMNAPOLB
SCHEMBL316461 0.76 KCNH2 (0.44) ALDH1A1MAPTLMNAPOLB
SCHEMBL1402778 0.75 HSD11B1 (0.72) ALDH1A1MAPTMAPK1GAALMNA
SCHEMBL2987752 0.75 CNR2 (0.42) ALDH1A1MAPTLMNAPOLB
SCHEMBL315723 0.75 ALDH1A1 (0.54) ALDH1A1MAPTMAPK1GAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US claimed
US-8093272-B2 Heteroaryl substituted cyclohexyl-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2012-01-10 US disclosed