SCHEMBL3173519

SCHEMBL3173519

c1ccc(Cc2ccc([C](c3ccccc3)c3ccccc3)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CALM1 P0DP23 1/20 0.60
LMNA P02545 2/20 0.59
PLA2G10 O15496 1/20 0.59
PLA2G2A P14555 1/20 0.59
IDH1 O75874 1/20 0.50
PRSS1 P07477 1/20 0.48
PRSS2 P07478 1/20 0.48
PRSS3 P35030 1/20 0.48
SRD5A2 P31213 1/20 0.47
SLC22A2 O15244 1/20 0.47
LTA4H P09960 1/20 0.46
KMT2A Q03164 1/20 0.44
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
BCL2 P10415 1/20 0.43
BCL2L1 Q07817 1/20 0.43
TSHR P16473 2/20 0.42
CYP2C9 P11712 1/20 0.42
HNF4A P41235 1/20 0.42
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Thiobenzoic Acid SCHEMBL29060734 0.81 LMNA (0.55) CALM1LMNAPLA2G10PLA2G2AIDH1
SCHEMBL9806315 0.81 LMNA (0.55) CALM1LMNAPLA2G10PLA2G2AIDH1
SCHEMBL7895911 0.81 LMNA (0.55) CALM1LMNAPLA2G10PLA2G2AIDH1
SCHEMBL4004691 0.81 LMNA (0.67) CALM1LMNAPLA2G10PLA2G2ASRD5A2
SCHEMBL8094422 0.81 CALM1 (0.92) CALM1LMNAPLA2G10PLA2G2AIDH1
Diphenylmethane SCHEMBL10394702 0.81 CALM1 (0.92) CALM1LMNAPLA2G10PLA2G2AIDH1
SCHEMBL972712 0.81 CALM1 (0.92) CALM1LMNAPLA2G10PLA2G2AIDH1
SCHEMBL14361865 0.78 TP53 (0.59) LMNACES2CES1
SCHEMBL5482345 0.78 SRD5A2 (0.71) CALM1LMNAPLA2G10PLA2G2ASRD5A2
Benzoic Acid SCHEMBL7064148 0.78 SRD5A2 (0.71) LMNAPLA2G10PLA2G2ASRD5A2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105693817-B Tripeptide compound and preparation method and application thereof 西北大学 2020-06-05 CN disclosed
CN-105693817-A Tripeptide compound and preparation method and application thereof 西北大学 2016-06-22 CN disclosed
WO-2013181697-A1 BICYCLO[6.1.0]NON-4-YNE COMPOUNDS SUITABLE FOR USE AS LINKERS IN BIOLOGICAL APPLICATIONS THE UNIVERSITY OF MELBOURNE (AU) 2013-12-12 WO disclosed
US-8298513-B2 Hexatriene-β-carbonyl compound OSAKA UNIVERSITY (JP) 2012-10-30 US disclosed
US-20100008857-A1 NOVEL HEXATRIENE-BETA-CARBONYL COMPOUND OSAKA UNIVERSITY (JP) 2010-01-14 US disclosed
CN-1198833-C Acetyl pyrrolidone cephlosporins with basic substitutent group BASILEA PHARMACEUTICA AG (CH) 2005-04-27 CN disclosed
US-RE36374-E 1,2,3-triazole and tetrazole substituted piperidine or tetrahydropyridine compounds useful as acetylcholine agonists H. LUNDBECK, A/S (DK) 1999-11-02 US disclosed
US-5972929-A Quinazolinone derivative, hair growth promoter and external composition for skin using the same SHISEIDO CO., LTD. (JP) 1999-10-26 US disclosed
EP-0296721-B1 HETEROCYCLIC COMPOUNDS H. LUNDBECK A/S (DK) 1993-06-23 EP disclosed
US-4925858-A NERVOUS SYSTEM DISORDERS, ALZHEIMER*S DISEASE H. LUNDBECK A/S (DK) 1990-05-15 US disclosed
US-4866077-A TREATMENT OF NERVOUS SYSTEM DISORDERS SUCH AS ALZHEIMER*S DISEASE H. LUNDBECK A/S (DK) 1989-09-12 US disclosed
EP-0296721-A2 Heterocyclic compounds H. LUNDBECK A/S (DK) 1988-12-28 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100008857-A1 NOVEL HEXATRIENE-BETA-CARBONYL COMPOUND CBR1, CBR3, DCXR CALM1 2454/4885LMNA 2666/4885PLA2G10 3873/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.