SCHEMBL3188564

SCHEMBL3188564

C#C[C@H]1CCCN1C(=O)OC(C)(C)C

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.55
HPGD P15428 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.45
ALDH1A1 P00352 2/20 0.44
MEN1 O00255 1/20 0.44
MAPT P10636 1/20 0.44
KMT2A Q03164 1/20 0.44
CTSK P43235 1/20 0.43
NPC1 O15118 1/20 0.42
RECQL P46063 1/20 0.42
LMNA P02545 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL231219 1.00 HSD17B10 (0.55) HSD17B10HPGDSMN1; SMN2ALDH1A1MEN1
SCHEMBL889059 1.00 HSD17B10 (0.55) HSD17B10HPGDSMN1; SMN2ALDH1A1MEN1
SCHEMBL525478 0.95 HPGD (0.50) HSD17B10HPGDSMN1; SMN2ALDH1A1MEN1
SCHEMBL10082580 0.95 HPGD (0.50) HSD17B10HPGDSMN1; SMN2ALDH1A1MEN1
SCHEMBL15317053 0.95 HPGD (0.50) HSD17B10HPGDSMN1; SMN2ALDH1A1MEN1
SCHEMBL5275535 0.90 HSD17B10 (0.47) HSD17B10HPGDSMN1; SMN2ALDH1A1MEN1
SCHEMBL4919669 0.90 HSD17B10 (0.47) HSD17B10HPGDSMN1; SMN2ALDH1A1MEN1
SCHEMBL29530476 0.89 HSD17B10 (0.46) HSD17B10HPGDSMN1; SMN2ALDH1A1MEN1
SCHEMBL1198458 0.87 PTPN2 (0.47) HSD17B10HPGDNPC1LMNANPSR1
SCHEMBL5171011 0.85 HSD17B10 (0.49) HSD17B10HPGDSMN1; SMN2ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 89 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260078121-A1 INHIBITORS OF ENL/AF9 YEATS AND FLT3 BRIDGE MEDICINES (US) 2026-03-19 US disclosed
WO-2025262297-A1 PROTAC DEGRADERS OF MLLT1 AND/OR MLLT3 DARK BLUE THERAPEUTICS LTD (GB) 2025-12-26 WO disclosed
WO-2025262295-A1 PROTAC DEGRADERS OF MLLT1 AND/OR MLLT3 DARK BLUE THERAPEUTICS LTD (GB) 2025-12-26 WO disclosed
EP-4667466-A1 PROTAC DEGRADERS OF MLLT1 AND/OR MLLT3 Dark Blue Therapeutics Ltd (GB) 2025-12-24 EP disclosed
EP-4667467-A1 PROTAC DEGRADERS OF MLLT1 AND/OR MLLT3 Dark Blue Therapeutics Ltd (GB) 2025-12-24 EP disclosed
US-20250368641-A1 QUINOLINE COMPOUNDS AS INHIBITORS OF KRAS INCYTE CORP (US) 2025-12-04 US disclosed
US-12378243-B2 Quinoline compounds as inhibitors of KRAS INCYTE CORPORATION (US) 2025-08-05 US disclosed
EP-4583869-A2 INHIBITORS OF ENL/AF9 YEATS AND FLT3 Bridge Medicines (US) 2025-07-16 EP disclosed
WO-2025111492-A1 INHIBITORS OF PARG 858 THERAPEUTICS, INC. (US) 2025-05-30 WO disclosed
US-20250171402-A1 Potent and Selective Human Neuronal Nitric Oxide Synthase Inhibitors UNIV NORTHWESTERN (US) 2025-05-29 US disclosed
EP-0440670-B1 HETEROCYCLIC ACETYLENIC AMINES HAVING CENTRAL NERVOUS SYSTEM ACTIVITY UPJOHN CO (US) 1996-03-06 EP disclosed
US-5409946-A Antiepileptic agent ABBOTT LABORATORIES (US) 1995-04-25 US disclosed
EP-0588917-A4 1994-04-13 EP disclosed
EP-0588917-A1 ISOXAZOLE AND ISOTHIAZOLE COMPOUNDS THAT ENHANCE COGNITIVE FUNCTION ABBOTT LABORATORIES (US) 1994-03-30 EP disclosed
US-5225567-A HETEROCYCLIC ACETYLENIC AMINES HAVING CENTRAL NERVOUS SYSTEM ACTIVITY THE UPJOHN COMPANY (US) 1993-07-06 US disclosed
WO-1992021339-A1 ISOXAZOLE AND ISOTHIAZOLE COMPOUNDS THAT ENHANCE COGNITIVE FUNCTION ABBOTT LABORATORIES (US) 1992-12-10 WO disclosed
US-5157124-A Improving mental performance THE UPJOHN COMPANY (US) 1992-10-20 US disclosed
US-5137905-A Cholinergic agonists; analgesics; cognition activators THE UPJOHN COMPANY (US) 1992-08-11 US disclosed
EP-0440670-A1 HETEROCYCLIC ACETYLENIC AMINES HAVING CENTRAL NERVOUS SYSTEM ACTIVITY. UPJOHN CO (US) 1991-08-14 EP disclosed
WO-1990004588-A1 HETEROCYCLIC ACETYLENIC AMINES HAVING CENTRAL NERVOUS SYSTEM ACTIVITY THE UPJOHN COMPANY (US) 1990-05-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12378243-B2 Quinoline compounds as inhibitors of KRAS KRAS, NRAS, HRAS HSD17B10 3790/4885HPGD 647/4885SMN1; SMN2 3339/4885
US-20250368641-A1 QUINOLINE COMPOUNDS AS INHIBITORS OF KRAS KRAS, NRAS, HRAS HSD17B10 3790/4885HPGD 647/4885SMN1; SMN2 3339/4885
US-20250171402-A1 Potent and Selective Human Neuronal Nitric Oxide Synthase Inhibitors NOS2, NOS1, NOS3 HSD17B10 1278/4885HPGD 13/4885SMN1; SMN2 71/4885
US-20260078121-A1 INHIBITORS OF ENL/AF9 YEATS AND FLT3 MLLT3, MLLT1, FLT3 HSD17B10 2268/4885HPGD 4318/4885SMN1; SMN2 4179/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.