SCHEMBL3194786

SCHEMBL3194786

COc1cc(/C=C/C(=O)/C=C/c2ccc(OCC(=O)O)c(OC)c2)ccc1OCC(=O)O

nearest known ligand 0.85

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.85
HDAC2 Q92769 1/20 0.85
HDAC8 Q9BY41 1/20 0.85
POLB P06746 1/20 0.77
APP P05067 4/20 0.73
SNCA P37840 1/20 0.67
NFKB1 P19838 2/20 0.63
JUN P05412 1/20 0.63
FDPS P14324 3/20 0.62
KDM4E B2RXH2 2/20 0.61
ALDH1A1 P00352 2/20 0.61
HPGD P15428 1/20 0.61
ALOX15 P16050 1/20 0.61
MAPK1 P28482 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
HSD17B10 Q99714 1/20 0.61
NFE2L2 Q16236 2/20 0.60
CYP1A2 P05177 1/20 0.60
ALOX5 P09917 1/20 0.60
CYP2D6 P10635 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3194804 1.00 HDAC1 (0.85) HDAC1HDAC2HDAC8POLBAPP
SCHEMBL25275685 0.91 SNCA (0.80) HDAC1HDAC2HDAC8POLBAPP
SCHEMBL19918301 0.91 SNCA (0.80) HDAC1HDAC2HDAC8POLBAPP
SCHEMBL14887104 0.90 APP (0.88) HDAC1HDAC2HDAC8POLBAPP
SCHEMBL16868836 0.90 APP (0.88) HDAC1HDAC2HDAC8POLBAPP
SCHEMBL5429268 0.89 FDPS (0.78) HDAC1HDAC2HDAC8POLBAPP
SCHEMBL5429269 0.89 FDPS (0.78) HDAC1HDAC2HDAC8POLBAPP
SCHEMBL25189341 0.85 MAPT (0.80) HDAC1HDAC2HDAC8POLBAPP
SCHEMBL25265169 0.85 MAPT (0.80) HDAC1HDAC2HDAC8POLBAPP
SCHEMBL2743877 0.85 NFKB1 (0.79) NFKB1JUNKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100029763-A1 METHODS TO PREPARE PENTA-1,4-DIEN-3-ONES AND SUBSTITUTED CYCLOHEXANONES AND DERIVATIVES WITH ANTITUMORAL AND ANTIPARASITIC PROPERTIES, THE COMPOUNDS AND THEIR USES UNIVERSIDADE BANDEIRANTE DE SAO PAULO-ACADEMIA, PAULISTA ANCHIETA S/C LTDA (BR) 2010-02-04 US claimed
EP-2054365-A2 METHODS TO PREPARE PENTA-1,4-DIEN-3-ONES AND SUBSTITUTED CYCLOHEXANONES AND DERIVATIVES WITH ANTITUMORAL AND ANTIPARASITIC PROPERTIES, THE COMPOUNDS AND THEIR USES Uniban - Universidade Bandeirante De São Paulo (BR) 2009-05-06 EP claimed
WO-2008003155-A2 METHODS TO PREPARE PENTA-1,4-DIEN-3-ONES AND SUBSTITUTED CYCLOHEXANONES AND DERIVATIVES WITH ANTITUMORAL AND ANTIPARASITIC PROPERTIES, THE COMPOUNDS AND THEIR USES UNIBAN - UNIVERSIDADE BANDEIRANTE DE SÃO PAULO - ACADEMIA PAULISTA ANCHIETA S/C LTDA (BR) 2008-01-10 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100029763-A1 METHODS TO PREPARE PENTA-1,4-DIEN-3-ONES AND SUBSTITUTED CYCLOHEXANONES AND DERIVATIVES WITH ANTITUMORAL AND ANTIPARASITIC PROPERTIES, THE COMPOUNDS AND THEIR USES CASP3, CYP8B1, DERA HDAC1 2278/4885HDAC2 2823/4885HDAC8 3304/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.