Alacepril

Alacepril

SCHEMBL3204613

CC(=O)SCC(C)C(=O)N1CCC[C@@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)O

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACE P12821 9/20 0.55
SLC6A2 P23975 1/20 0.54
ACE2 Q9BYF1 4/20 0.54
CMA1 P23946 2/20 0.53
OPRM1 P35372 1/20 0.51
DPP3 Q9NY33 1/20 0.50
ALDH1A1 P00352 1/20 0.50
HSD17B10 Q99714 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Alacepril SCHEMBL11460465 1.00 ACE (0.55) ACESLC6A2ACE2CMA1OPRM1
Alacepril SCHEMBL5058556 1.00 ACE (0.55) ACESLC6A2ACE2CMA1OPRM1
Alacepril SCHEMBL20126832 1.00 ACE (0.55) ACESLC6A2ACE2CMA1OPRM1
Alacepril SCHEMBL683027 1.00 ACE (0.55) ACESLC6A2ACE2CMA1OPRM1
Alacepril SCHEMBL34559 1.00 ACE (0.55) ACESLC6A2ACE2CMA1OPRM1
Alacepril SCHEMBL28035498 1.00 ACE (0.55) ACESLC6A2ACE2CMA1OPRM1
Alacepril SCHEMBL677447 1.00 ACE (0.55) ACESLC6A2ACE2CMA1OPRM1
Alacepril SCHEMBL11458085 0.95 ACE (0.51) ACESLC6A2ACE2CMA1OPRM1
SCHEMBL11282561 0.93 SLC6A2 (0.56) ACESLC6A2CMA1OPRM1
SCHEMBL683119 0.93 SLC6A2 (0.56) ACESLC6A2CMA1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-11222439-A None JP disclosed
EP-2198869-B1 TREHALOSE FOR THE TREATMENT OR PREVENTION OF VASOSPASM NEXT 21 K K (JP) 2015-09-16 EP disclosed
US-8283337-B2 Therapeutic or prophylactic agent for vasoconstriction NEXT21 K.K. (JP) 2012-10-09 US disclosed
EP-2198869-A1 THERAPEUTIC OR PROPHYLACTIC AGENT FOR VASOCONSTRICTION Next 21 K.K. (JP) 2010-06-23 EP disclosed
US-20100035837-A1 THERAPEUTIC OR PROPHYLACTIC AGENT FOR VASOCONSTRICTION NEXT21 K.K. (JP) 2010-02-11 US disclosed
EP-1323434-B1 Method for diagnostic imaging of the renal region using a contrast agent and a vasodilator IMARX PHARMACEUTICAL CORP (US) 2007-07-11 EP disclosed
EP-1323434-A2 Improved methods for diagnostic imaging using a contrast agent and a vasodilator IMARX PHARMACEUTICAL CORP. (US) 2003-07-02 EP disclosed
EP-0977597-B1 IMPROVED METHODS FOR DIAGNOSTIC IMAGING USING A CONTRAST AGENT AND A VASODILATOR IMARX PHARMACEUTICAL CORP (US) 2003-01-15 EP disclosed
US-6071494-A LIPID, PROTEIN OR POLYMER AND A GAS OR GASEOUS PRECURSOR, IN COMBINATION WITH A RENAL VASODILATOR. IMARX PHARMACEUTICAL CORP. (US) 2000-06-06 US disclosed
JP-H11222439-A INHIBITOR OF CEREBRAL VASOSPASM DAINIPPON PHARMACEUT CO LTD 1999-08-17 JP disclosed