Alacepril

Alacepril

SCHEMBL677447

CC(=O)SCC(C)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)O

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACE P12821 9/20 0.55
SLC6A2 P23975 1/20 0.54
ACE2 Q9BYF1 4/20 0.54
CMA1 P23946 2/20 0.53
OPRM1 P35372 1/20 0.51
DPP3 Q9NY33 1/20 0.50
ALDH1A1 P00352 1/20 0.50
HSD17B10 Q99714 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Alacepril SCHEMBL11460465 1.00 ACE (0.55) ACESLC6A2ACE2CMA1OPRM1
Alacepril SCHEMBL5058556 1.00 ACE (0.55) ACESLC6A2ACE2CMA1OPRM1
Alacepril SCHEMBL20126832 1.00 ACE (0.55) ACESLC6A2ACE2CMA1OPRM1
Alacepril SCHEMBL683027 1.00 ACE (0.55) ACESLC6A2ACE2CMA1OPRM1
Alacepril SCHEMBL34559 1.00 ACE (0.55) ACESLC6A2ACE2CMA1OPRM1
Alacepril SCHEMBL3204613 1.00 ACE (0.55) ACESLC6A2ACE2CMA1OPRM1
Alacepril SCHEMBL28035498 1.00 ACE (0.55) ACESLC6A2ACE2CMA1OPRM1
Alacepril SCHEMBL11458085 0.95 ACE (0.51) ACESLC6A2ACE2CMA1OPRM1
SCHEMBL11282561 0.93 SLC6A2 (0.56) ACESLC6A2CMA1OPRM1
SCHEMBL683119 0.93 SLC6A2 (0.56) ACESLC6A2CMA1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0007477-B1 1-(3-MERCAPTO-2-METHYLPROPANOYL)PROLYL AMINO ACID DERIVATIVES AND SALTS THEREOF, PROCESSES FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH COMPOUNDS Dainippon Pharmaceutical Co., Ltd. (JP) 1982-04-28 EP claimed
US-4248883-A ANTIHYPERTENSION AGENTS DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1981-02-03 US claimed
EP-0007477-A1 1-(3-Mercapto-2-methylpropanoyl)prolyl amino acid derivatives and salts thereof, processes for their preparation, and pharmaceutical compositions containing such compounds Dainippon Pharmaceutical Co., Ltd. (JP) 1980-02-06 EP claimed
JP-11222439-A None JP disclosed
JP-56092848-A None JP disclosed
JP-56145220-A None JP disclosed
EP-2198869-B1 TREHALOSE FOR THE TREATMENT OR PREVENTION OF VASOSPASM NEXT 21 K K (JP) 2015-09-16 EP disclosed
US-8283337-B2 Therapeutic or prophylactic agent for vasoconstriction NEXT21 K.K. (JP) 2012-10-09 US disclosed
US-20110269717-A1 NEUROGENESIS BY MODULATING ANGIOTENSIN BRAINCELLS INC. (US) 2011-11-03 US disclosed
EP-2382975-A2 Neurogenesis by modulating angiotensin Braincells, Inc. (US) 2011-11-02 EP disclosed
EP-2377531-A2 Neurogenesis by modulating angiotensin Braincells, Inc. (US) 2011-10-19 EP disclosed
US-5846517-A Methods for diagnostic imaging using a renal contrast agent and a vasodilator IMARX PHARMACEUTICAL CORP. (US) 1998-12-08 US disclosed
EP-0105696-B1 OPTICALLY ACTIVE N-SUBSTITUTED PHENYLALANINOLS AND USE THEREFOR Dainippon Pharmaceutical Co., Ltd. (JP) 1986-01-02 EP disclosed
US-4536601-A USE FOR RESOLUTION OF D-3-ACETHYLTHIO-2-METHYLPROPIONIC ACID DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1985-08-20 US disclosed
EP-0105696-A1 Optically active N-substituted phenylalaninols and use therefor Dainippon Pharmaceutical Co., Ltd. (JP) 1984-04-18 EP disclosed
EP-0007477-B1 1-(3-MERCAPTO-2-METHYLPROPANOYL)PROLYL AMINO ACID DERIVATIVES AND SALTS THEREOF, PROCESSES FOR THEIR PREPARATION, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SUCH COMPOUNDS Dainippon Pharmaceutical Co., Ltd. (JP) 1982-04-28 EP disclosed
JP-S56145220-A ANTIHYPERTENSIVE AGENT CONTAINING PROLYLAMINO ACID DERIVATIVE AND DIURETIC AGENT AS MAIN CONSTITUENT DAINIPPON PHARMACEUT CO LTD 1981-11-11 JP disclosed
JP-S5692848-A PREPARATION OF 1- 3-LOWER ALAKNOYLTHIO-2-METHYLPROPANOYL PROLYLPHENYLALANINE DAINIPPON PHARMACEUT CO LTD 1981-07-27 JP disclosed
US-4248883-A ANTIHYPERTENSION AGENTS DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1981-02-03 US disclosed
EP-0007477-A1 1-(3-Mercapto-2-methylpropanoyl)prolyl amino acid derivatives and salts thereof, processes for their preparation, and pharmaceutical compositions containing such compounds Dainippon Pharmaceutical Co., Ltd. (JP) 1980-02-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110269717-A1 NEUROGENESIS BY MODULATING ANGIOTENSIN NGF, DCX, BDNF ACE 6/4885SLC6A2 376/4885ACE2 11/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.