SCHEMBL3207282

SCHEMBL3207282

O=C(O)/C=C/c1ccc(O)cc1OCc1ccccc1

nearest known ligand 0.70

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 5/20 0.70
PTGER2 P43116 5/20 0.70
PTGER3 P43115 5/20 0.70
PTGER1 P34995 4/20 0.70
HDAC8 Q9BY41 1/20 0.57
BACE1 P56817 1/20 0.55
KDM4E B2RXH2 2/20 0.54
LMNA P02545 1/20 0.54
AKR1B10 O60218 2/20 0.54
AKR1B1 P15121 2/20 0.54
ALDH1A1 P00352 1/20 0.53
PKM P14618 1/20 0.53
MIF P14174 1/20 0.51
PTGDR Q13258 1/20 0.51
LTB4R Q15722 1/20 0.51
LTB4R2 Q9NPC1 1/20 0.51
APP P05067 1/20 0.50
AKR1C3 P42330 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3207292 1.00 PTGER4 (0.70) PTGER4PTGER2PTGER3PTGER1HDAC8
SCHEMBL344776 0.89 PTGER4 (0.70) PTGER4PTGER2PTGER3PTGER1HDAC8
SCHEMBL344775 0.89 PTGER4 (0.70) PTGER4PTGER2PTGER3PTGER1HDAC8
SCHEMBL7191225 0.87 PTGER3 (0.68) PTGER4PTGER2PTGER3PTGER1HDAC8
SCHEMBL7909151 0.87 PTGER3 (0.68) PTGER4PTGER2PTGER3PTGER1HDAC8
SCHEMBL9199949 0.87 HDAC8 (0.65) PTGER4PTGER2PTGER3PTGER1HDAC8
SCHEMBL3409441 0.86 PTGER4 (0.67) PTGER4PTGER2PTGER3PTGER1HDAC8
SCHEMBL3409444 0.86 PTGER4 (0.67) PTGER4PTGER2PTGER3PTGER1HDAC8
SCHEMBL8323200 0.85 PTGER4 (0.94) PTGER4PTGER2PTGER3PTGER1HDAC8
SCHEMBL8323198 0.85 PTGER4 (0.94) PTGER4PTGER2PTGER3PTGER1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100041892-A1 Therapeutic agent for diabetes ABE HIDENORI 2010-02-18 US disclosed
US-20090270631-A1 Therapeutic agent for diabetes ABE HIDENORI 2009-10-29 US disclosed
EP-1912645-A2 THERAPEUTIC AGENT FOR DIABETES Takeda Pharmaceutical Company Limited (JP) 2008-04-23 EP disclosed
US-20080051418-A1 Arylalkanoic Acid Derivative TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-02-28 US disclosed
US-20080009530-A1 Therapeutic Agent for Diabetes TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-01-10 US disclosed
EP-1829863-A1 ARYLALKANOIC ACID DERIVATIVE Takeda Pharmaceutical Company Limited (JP) 2007-09-05 EP disclosed
WO-2007018314-A2 THERAPEUTIC AGENT FOR DIABETES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090270631-A1 Therapeutic agent for diabetes FABP4, SLC5A1, SLC5A2 PTGER4 2014/4885PTGER2 2887/4885PTGER3 2459/4885
US-20080051418-A1 Arylalkanoic Acid Derivative INSR, NPY1R, GPR119 PTGER4 1928/4885PTGER2 3643/4885PTGER3 1565/4885
US-20080009530-A1 Therapeutic Agent for Diabetes FABP4, SLC5A1, SLC5A2 PTGER4 2098/4885PTGER2 2361/4885PTGER3 2522/4885
US-20100041892-A1 Therapeutic agent for diabetes FABP4, SLC5A1, SLC5A2 PTGER4 2014/4885PTGER2 2887/4885PTGER3 2459/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.