SCHEMBL3215218

SCHEMBL3215218

O=C(NC(CCc1ccccc1)C(=O)NC(CCc1ccccc1)C(=O)O)c1ccc(Cl)c(-c2ccc(-c3ccccc3)cc2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 2/20 0.52
PDK2 Q15119 2/20 0.52
PDK3 Q15120 2/20 0.52
PDK4 Q16654 2/20 0.52
CA1 P00915 4/20 0.47
CA2 P00918 4/20 0.47
MME P08473 2/20 0.47
ACE P12821 1/20 0.47
CPA1 P15085 1/20 0.47
ACE2 Q9BYF1 1/20 0.47
ERAP2 Q6P179 1/20 0.45
ERAP1 Q9NZ08 1/20 0.45
LNPEP Q9UIQ6 1/20 0.45
GPR132 Q9UNW8 2/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
CTSL P07711 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3199823 0.89 PDK1 (0.53) PDK1PDK2PDK3PDK4CA1
SCHEMBL3222613 0.88 GRN (0.51) PDK1PDK2PDK3PDK4MME
SCHEMBL3213081 0.88 GPR132 (0.50) PDK1PDK2PDK3PDK4CA1
SCHEMBL3218617 0.86 PDK1 (0.42) PDK1PDK2PDK3PDK4CA1
SCHEMBL3222001 0.86 GPR132 (0.55) PDK1PDK2PDK3PDK4GPR132
SCHEMBL775117 0.81 CA2 (0.64) CA1CA2MEN1KMT2ACYP1A2
SCHEMBL18653875 0.77 LNPEP (0.52) PDK1PDK2PDK3PDK4ERAP2
SCHEMBL15989069 0.77 LNPEP (0.52) PDK1PDK2PDK3PDK4ERAP2
SCHEMBL775213 0.77 GRN (0.59) PDK1PDK2PDK3PDK4CA1
SCHEMBL3215269 0.75 PDK1 (0.52) PDK1PDK2PDK3PDK4CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7683097-B2 Topoisomerase inhibitors Propharmacon Inc. (US) 2010-03-23 US claimed