SCHEMBL321580

SCHEMBL321580

COC(=O)c1cccc(OCCC(=O)OCc2ccccc2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.53
MRGPRX4 Q96LA9 1/20 0.53
ALDH1A1 P00352 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
NR4A2 P43354 1/20 0.52
SMPD1 P17405 1/20 0.51
MAPT P10636 2/20 0.50
RAB9A P51151 2/20 0.50
CYSLTR1 Q9Y271 1/20 0.49
HPGD P15428 2/20 0.49
PTPN1 P18031 1/20 0.49
LMNA P02545 1/20 0.49
MEN1 O00255 1/20 0.48
POLB P06746 1/20 0.48
KMT2A Q03164 1/20 0.48
KDM4E B2RXH2 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25364811 0.86 ALDH1A1 (0.57) MAOBMRGPRX4ALDH1A1CYP1A2CYP3A4
SCHEMBL29524175 0.86 ALDH1A1 (0.57) MAOBMRGPRX4ALDH1A1CYP1A2CYP3A4
SCHEMBL30412034 0.84 MAOB (0.73) MAOBMRGPRX4NR4A2SMPD1CYSLTR1
SCHEMBL976424 0.84 MAOB (0.73) MAOBMRGPRX4NR4A2SMPD1CYSLTR1
SCHEMBL24627608 0.83 L3MBTL1 (0.65) MAOBMRGPRX4ALDH1A1CYP1A2CYP3A4
SCHEMBL3538378 0.82 L3MBTL1 (0.61) MAOBMRGPRX4ALDH1A1CYP1A2CYP3A4
SCHEMBL1122805 0.82 MRGPRX4 (0.71) MAOBMRGPRX4NR4A2SMPD1CYSLTR1
SCHEMBL320846 0.82 ALDH1A1 (0.59) MRGPRX4ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL11401546 0.81 ALDH1A1 (0.58) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL1122722 0.81 MAOB (0.68) MAOBMRGPRX4NR4A2SMPD1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2590942-A1 RHO KINASE INHIBITORS Boehringer Ingelheim International GmbH (DE) 2013-05-15 EP disclosed
WO-2012006202-A1 RHO KINASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-01-12 WO disclosed