SCHEMBL3226086

SCHEMBL3226086

C=CCN(CC=C)c1c[nH]nn1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8722271 0.69 ALDH1A1 (0.39)
SCHEMBL232139 0.68
SCHEMBL622400 0.68
SCHEMBL4724612 0.67 HCAR3 (0.33)
SCHEMBL2226753 0.66
SCHEMBL951386 0.64
SCHEMBL22372230 0.64 SCN9A (0.36)
SCHEMBL11729624 0.63 ALDH1A1 (0.32)
SCHEMBL4550661 0.63
SCHEMBL9472234 0.63 CRHR1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2391631-B1 NOVEL MATERIAL WITH SPIN TRANSITION, AND METHOD FOR MAKING SAME CENTRE NAT RECH SCIENT (FR) 2015-03-11 EP disclosed
EP-2170915-B1 SPIN TRANSITION MATERIAL CENTRE NAT RECH SCIENT (FR) 2015-01-14 EP disclosed
US-8753743-B2 Nanoparticles of a spin transition compound CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2014-06-17 US disclosed
US-8709599-B2 Spin transition material CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2014-04-29 US disclosed
US-20130011680-A1 NANOPARTICLES OF A SPIN TRANSITION COMPOUND CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2013-01-10 US disclosed
EP-2391631-A1 NOVEL MATERIAL WITH SPIN TRANSITION, AND METHOD FOR MAKING SAME Centre National de la Recherche Scientifique (FR) 2011-12-07 EP disclosed
WO-2010086550-A1 NOVEL MATERIAL WITH SPIN TRANSITION, AND METHOD FOR MAKING SAME CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2010-08-05 WO disclosed
US-20100178511-A1 SPIN TRANSITION MATERIAL CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2010-07-15 US disclosed
EP-2170915-A2 SPIN TRANSITION MATERIAL Centre National De La Recherche Scientifique (FR) 2010-04-07 EP disclosed
EP-1960410-B1 NANOPARTICLES OF A SPIN TRANSITION COMPOUND CENTRE NAT RECH SCIENT (FR) 2010-03-03 EP disclosed
WO-2009007534-A2 SPIN TRANSITION MATERIAL CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2009-01-15 WO disclosed
US-20080311401-A1 Nanoparticle of a Spin Transition Compound CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2008-12-18 US disclosed
EP-1960410-A1 NANOPARTICLES OF A SPIN TRANSITION COMPOUND Centre National de la Recherche Scientifique (FR) 2008-08-27 EP disclosed
WO-2007065996-A1 NANOPARTICLES OF A SPIN TRANSITION COMPOUND CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2007-06-14 WO disclosed