SCHEMBL323013

SCHEMBL323013

CCCn1c(=O)[nH]c2ccc(C(=O)c3ncc4ccc(C(=O)OC(=O)c5ccc6cnc(C(=O)c7ccc(N)c(C(=O)O)c7)n6c5)cn34)cc2c1=O

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.37
GAA P10253 7/20 0.37
ALDH1A1 P00352 6/20 0.37
HSD17B10 Q99714 4/20 0.37
HPGD P15428 3/20 0.37
POLB P06746 2/20 0.35
HPD P32754 4/20 0.33
GLA P06280 3/20 0.33
KMT2A Q03164 2/20 0.33
PKM P14618 1/20 0.33
HTT P42858 1/20 0.33
HTR3A P46098 1/20 0.33
ADORA3 P0DMS8 2/20 0.32
ADORA2B P29275 2/20 0.32
TP53 P04637 2/20 0.32
MAPT P10636 2/20 0.32
ADORA1 P30542 1/20 0.32
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL323012 0.95 KDM4E (0.42) KDM4EGAAALDH1A1HSD17B10HPGD
SCHEMBL321649 0.87 KDM4E (0.48) KDM4EGAAALDH1A1HSD17B10HPGD
SCHEMBL17074451 0.82 KDM4E (0.39) KDM4EGAAALDH1A1HSD17B10HPGD
SCHEMBL17074452 0.81 KDM4E (0.39) KDM4EGAAALDH1A1HSD17B10HPGD
SCHEMBL327753 0.77 KDM4E (0.41) KDM4EGAAALDH1A1HSD17B10HPGD
SCHEMBL321841 0.74 MAPT (0.42) KDM4EGAAALDH1A1HSD17B10POLB
SCHEMBL321406 0.70 KDM4E (0.44) KDM4EGAAALDH1A1HSD17B10HPGD
SCHEMBL323368 0.68 NPC1 (0.43) KDM4EGAAALDH1A1HSD17B10HPGD
SCHEMBL322028 0.67 MAPK8 (0.34) KDM4EGAAALDH1A1HSD17B10HPGD
SCHEMBL14927289 0.65 ADORA3 (0.43) KDM4EALDH1A1HSD17B10HPGDHPD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2590976-A1 IMIDAZOPYRIDINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2013-05-15 EP disclosed
WO-2012004732-A1 IMIDAZOPYRIDINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI (FR) 2012-01-12 WO disclosed