SCHEMBL3230845

SCHEMBL3230845

CCCCP(=O)(Oc1ccccc1Cl)c1ccccc1Cl

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
PKM P14618 1/20 0.40
HSD17B10 Q99714 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TSHR P16473 2/20 0.39
PTK2B Q14289 1/20 0.38
POLB P06746 1/20 0.37
GAA P10253 1/20 0.37
HIF1A Q16665 1/20 0.36
HPGD P15428 2/20 0.36
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4422355 0.81 LMNA (0.51) LMNASMN1; SMN2PKML3MBTL1TSHR
SCHEMBL3226079 0.81 LMNA (0.51) LMNASMN1; SMN2PKML3MBTL1TSHR
SCHEMBL13430920 0.79 LMNA (0.49) LMNASMN1; SMN2PKML3MBTL1POLB
SCHEMBL3231499 0.77 LMNA (0.50) LMNASMN1; SMN2PKML3MBTL1POLB
SCHEMBL4426186 0.76 LMNA (0.49) LMNASMN1; SMN2PKM
SCHEMBL20067122 0.75 LMNA (0.45) LMNASMN1; SMN2PKML3MBTL1
SCHEMBL14216107 0.75 LMNA (0.45) LMNASMN1; SMN2PKML3MBTL1POLB
SCHEMBL11495536 0.73 THRA (0.47)
SCHEMBL30722828 0.73 PKM (0.51) LMNASMN1; SMN2PKML3MBTL1
SCHEMBL3238027 0.73 PKM (0.51) LMNASMN1; SMN2PKML3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180104263-A1 BUTYRYLCHOLINESTERASE INHIBITORS JAL THERAPEUTICS, LLC 2018-04-19 US disclosed
EP-2097428-B1 BUTYRYLCHOLINESTERASE INHIBITORS AND THEIR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES MGP BIOTECHNOLOGIES INC (US) 2018-02-28 EP disclosed
US-9757399-B2 Butyrylcholinesterase inhibitors JAL THERAPEUTICS, INC. (US) 2017-09-12 US disclosed
US-20160206635-A1 Butyrylcholinesterase Inhibitors JAL THERAPEUTICS, LLC 2016-07-21 US disclosed
US-20140073608-A1 Butyrylcholinesterase Inhibitors MGP BIOTECHNOLOGIES, LLC (US) 2014-03-13 US disclosed
US-20100069337-A1 BUTYRYLCHOLINESTERASE INHIBITORS JAL THERAPEUTICS, LLC 2010-03-18 US disclosed
EP-2097428-A2 BUTYRYLCHOLINESTERASE INHIBITORS AND THEIR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES Mgp Biotechnologies, Inc. (US) 2009-09-09 EP disclosed
WO-2008055249-A2 BUTYRYLCHOLINESTERASE INHIBITORS AND THEIR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES MGP BIOTECHNOLOGIES, INC. (US) 2008-05-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180104263-A1 BUTYRYLCHOLINESTERASE INHIBITORS BCHE, ACHE, PSEN1 LMNA 1641/4885SMN1; SMN2 178/4885PKM 746/4885
US-20160206635-A1 Butyrylcholinesterase Inhibitors BCHE, ACHE, PSEN1 LMNA 1641/4885SMN1; SMN2 178/4885PKM 746/4885
US-20140073608-A1 Butyrylcholinesterase Inhibitors BCHE, ACHE, PSEN1 LMNA 1641/4885SMN1; SMN2 178/4885PKM 746/4885
US-20100069337-A1 BUTYRYLCHOLINESTERASE INHIBITORS BCHE, ACHE, PSEN1 LMNA 1641/4885SMN1; SMN2 178/4885PKM 746/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.