SCHEMBL3237990

SCHEMBL3237990

Cc1cccc(C)c1C(=O)NC(c1ccccc1)C(C)(CO)N(C)C

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.47
SLC6A9 P48067 10/20 0.42
SLC6A5 Q9Y345 1/20 0.40
LMNA P02545 2/20 0.40
ITGB2 P05107 2/20 0.39
ICAM1 P05362 2/20 0.39
ITGAL P20701 2/20 0.39
UTS2R Q9UKP6 1/20 0.39
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CCR5 P51681 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3237956 0.91 L3MBTL1 (0.46) L3MBTL1SLC6A9SLC6A5LMNAITGB2
SCHEMBL3238003 0.86 UTS2R (0.47) LMNAUTS2RALDH1A1SMN1; SMN2
SCHEMBL3907148 0.85 SLC6A9 (0.47) L3MBTL1SLC6A9SLC6A5LMNAITGB2
SCHEMBL3240255 0.83 UTS2R (0.49) L3MBTL1SLC6A9LMNAITGB2ICAM1
SCHEMBL3239589 0.83 L3MBTL1 (0.40) L3MBTL1SLC6A9SLC6A5LMNAITGB2
SCHEMBL3238502 0.82 L3MBTL1 (0.47) L3MBTL1SLC6A9SLC6A5LMNAITGB2
SCHEMBL3238600 0.78 UTS2R (0.46) L3MBTL1LMNAUTS2RALDH1A1SMN1; SMN2
SCHEMBL3903930 0.78 SLC6A9 (0.41) L3MBTL1SLC6A9SLC6A5LMNAITGB2
SCHEMBL3906111 0.78 UTS2R (0.50) L3MBTL1SLC6A9LMNAITGB2ICAM1
SCHEMBL3905138 0.77 ATM (0.44) L3MBTL1SLC6A9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7745642-B2 Glycine transport inhibitors GLAXO GROUP LIMITED (GB) 2010-06-29 US disclosed
US-7745642-B2 Glycine transport inhibitors GLAXO GROUP LIMITED (GB) 2010-06-29 US disclosed
US-7745642-B2 Glycine transport inhibitors GLAXO GROUP LIMITED (GB) 2010-06-29 US disclosed
US-20080287547-A1 Glycine Transport Inhibitors GLAXO GROUP LIMITED (GB) 2008-11-20 US disclosed
US-20080287547-A1 Glycine Transport Inhibitors GLAXO GROUP LIMITED (GB) 2008-11-20 US disclosed
US-20080287547-A1 Glycine Transport Inhibitors GLAXO GROUP LIMITED (GB) 2008-11-20 US disclosed
WO-2006067423-A1 GLYCINE TRANSPORT INHIBITORS GLAXO GROUP LIMITED (GB) 2006-06-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080287547-A1 Glycine Transport Inhibitors SLC18A2, SLC6A5, SLC1A2 L3MBTL1 3944/4885SLC6A9 13/4885SLC6A5 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.