SCHEMBL3239589

SCHEMBL3239589

Cc1cccc(C)c1C(=O)NC(c1ccccc1)C(C)(CO[Si](C)(C)C(C)(C)C)N(C)C

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.40
SLC6A9 P48067 10/20 0.37
ITGB2 P05107 2/20 0.35
ICAM1 P05362 2/20 0.35
ITGAL P20701 2/20 0.35
SLC6A5 Q9Y345 1/20 0.35
UTS2R Q9UKP6 1/20 0.34
CCR5 P51681 2/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3243514 0.89 UTS2R (0.40) UTS2RLMNA
SCHEMBL3237990 0.83 L3MBTL1 (0.47) L3MBTL1SLC6A9ITGB2ICAM1ITGAL
SCHEMBL3237956 0.82 L3MBTL1 (0.46) L3MBTL1SLC6A9ITGB2ICAM1ITGAL
SCHEMBL3239756 0.79 CTSS (0.48) SLC6A9
SCHEMBL3907148 0.77 SLC6A9 (0.47) L3MBTL1SLC6A9ITGB2ICAM1ITGAL
SCHEMBL4358876 0.76 TACR3 (0.47)
SCHEMBL3240255 0.75 UTS2R (0.49) L3MBTL1SLC6A9ITGB2ICAM1ITGAL
SCHEMBL3238502 0.74 L3MBTL1 (0.47) L3MBTL1SLC6A9ITGB2ICAM1ITGAL
SCHEMBL3238003 0.71 UTS2R (0.47) UTS2RLMNA
SCHEMBL3905138 0.71 ATM (0.44) L3MBTL1SLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7745642-B2 Glycine transport inhibitors GLAXO GROUP LIMITED (GB) 2010-06-29 US disclosed
US-7745642-B2 Glycine transport inhibitors GLAXO GROUP LIMITED (GB) 2010-06-29 US disclosed
US-20080287547-A1 Glycine Transport Inhibitors GLAXO GROUP LIMITED (GB) 2008-11-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080287547-A1 Glycine Transport Inhibitors SLC18A2, SLC6A5, SLC1A2 L3MBTL1 3944/4885SLC6A9 13/4885ITGB2 4817/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.