SCHEMBL3242989

SCHEMBL3242989

CCCOC(=O)Oc1c[nH]c2c(=O)[nH]c3ccc(S(=O)(=O)[C@H]4CCC(N(C)C)C4)cc3c12

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.33
KDM4E B2RXH2 4/20 0.32
POLB P06746 2/20 0.31
MAPT P10636 2/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
HSD17B10 Q99714 4/20 0.31
MEN1 O00255 1/20 0.31
CYP2C9 P11712 1/20 0.31
KMT2A Q03164 1/20 0.31
MMP2 P08253 1/20 0.30
MMP9 P14780 1/20 0.30
MMP14 P50281 1/20 0.30
HPGD P15428 3/20 0.30
ALDH1A1 P00352 2/20 0.30
USP2 O75604 2/20 0.30
TSHR P16473 1/20 0.30
ESR1 P03372 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3254823 1.00 CASP3 (0.33) CASP3KDM4EPOLBMAPTLMNA
Hydrochloric Acid SCHEMBL3249857 0.88 CASP3 (0.33) CASP3KDM4EPOLBHSD17B10MEN1
Hydrochloric Acid SCHEMBL3252442 0.88 CASP3 (0.33) CASP3KDM4EPOLBHSD17B10MEN1
SCHEMBL3255160 0.86 MAPT (0.38) KDM4EPOLBMAPTLMNATP53
SCHEMBL3252606 0.84 ALDH1A1 (0.36) KDM4EPOLBMAPTLMNATP53
SCHEMBL3254901 0.83 KDM4E (0.38) CASP3KDM4EPOLBMAPTLMNA
SCHEMBL3245465 0.82 ALDH1A1 (0.36) KDM4EPOLBMAPTLMNATP53
SCHEMBL3243030 0.82 MAPT (0.34) KDM4EPOLBMAPTLMNATP53
SCHEMBL3251355 0.81 ALDH1A1 (0.37) KDM4EPOLBMAPTLMNATP53
SCHEMBL3251597 0.81 PARG (0.47) KDM4EPOLBMAPTLMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899335-B1 PYRROLOQUINOLINE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS PF MEDICAMENT (FR) 2010-05-19 EP claimed