SCHEMBL324349

SCHEMBL324349

NC(=O)c1ncccc1O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN2 Q96KS0 1/20 0.51
FTO Q9C0B1 1/20 0.51
KDM4E B2RXH2 5/20 0.49
TLR7 Q9NYK1 5/20 0.49
L3MBTL1 Q9Y468 4/20 0.45
ALDH1A1 P00352 3/20 0.45
TSHR P16473 3/20 0.45
MAPT P10636 3/20 0.45
CYP3A4 P08684 1/20 0.45
ALOX15 P16050 1/20 0.45
BLM P54132 1/20 0.45
AGER Q15109 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
HPGD P15428 1/20 0.45
HSD17B10 Q99714 1/20 0.45
PARP1 P09874 1/20 0.44
SPR P35270 1/20 0.44
THRB P10828 1/20 0.43
RAB9A P51151 1/20 0.43
MMP2 P08253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30452318 1.00 EGLN2 (0.51) EGLN2FTOKDM4ETLR7L3MBTL1
SCHEMBL27699633 0.82 FTO (0.55) EGLN2FTOKDM4ETLR7L3MBTL1
SCHEMBL518833 0.81 KDM4E (0.44) EGLN2FTOKDM4ETLR7L3MBTL1
SCHEMBL15312235 0.80 KDM4E (0.63) EGLN2FTOKDM4ETLR7L3MBTL1
SCHEMBL31356480 0.80 KDM4E (0.63) EGLN2FTOKDM4ETLR7L3MBTL1
SCHEMBL78249 0.80 KDM4E (0.63) EGLN2FTOKDM4ETLR7L3MBTL1
SCHEMBL4560363 0.80 MKNK1 (0.50) KDM4EL3MBTL1ALDH1A1TSHRMAPT
SCHEMBL8847897 0.80 EGLN2 (0.44) EGLN2FTOKDM4ETLR7L3MBTL1
SCHEMBL1985357 0.78 KDM4E (0.61) EGLN2FTOKDM4ETLR7L3MBTL1
SCHEMBL2277608 0.78 KDM4E (0.61) EGLN2FTOKDM4ETLR7L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 315 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220008414-A1 PHARMACEUTICAL COMPOSITION COMPRISING HISTONE DEACETYLASE 6 INHIBITORS CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2022-01-13 US claimed
US-10287255-B2 Compounds as histone deacetylase 6 inhibitors and pharmaceutical compositions comprising the same CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2019-05-14 US claimed
US-9932335-B2 Pyrrolopyridine or pyrazolopyridine derivatives HOFFMANN-LA ROCHE INC. (US) 2018-04-03 US claimed
US-20170096405-A1 NOVEL COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2017-04-06 US claimed
US-20160194321-A1 PYRROLOPYRIDINE OR PYRAZOLOPYRIDINE DERIVATIVES HOFFMANN-LA ROCHE INC. (US) 2016-07-07 US claimed
US-8735586-B2 Regioselective copper catalyzed synthesis of benzimidazoles and azabenzimidazoles SANOFI (FR) 2014-05-27 US claimed
US-8202834-B2 Fat regulation FIBROGEN, INC. (US) 2012-06-19 US claimed
EP-2173721-B1 A REGIOSELECTIVE COPPER CATALYZED SYNTHESIS OF BENZIMIDAZOLES AND AZABENZIMIDAZOLES SANOFI SA (FR) 2011-12-28 EP claimed
EP-2173747-B1 A REGIOSELECTIVE METAL CATALYZED SYNTHESIS OF ANNELATED BENZIMIDAZOLES AND AZABENZIMIDAZOLES SANOFI SA (FR) 2011-12-21 EP claimed
US-20110123434-A1 COMBINATION THERAPIES COMPRISING QUINOXALINE INHIBITORS OF P13K-ALPHA FOR USE IN THE TREATMENT OF CANCER EXELIXIS, INC (US) 2011-05-26 US claimed
WO-2006004507-A2 NEW BENZOTHIAZOLE DERIVATIVES USEFUL FOR TREATING CNS DISORDERS ASTRAZENECA AB (SE) 2006-01-12 WO claimed
US-20050155087-A1 Method of screening compounds NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2005-07-14 US claimed
EP-1463820-A1 METHOD OF SCREENING COMPOUNDS CHILDREN'S MEDICAL CENTER CORPORATION (US) 2004-10-06 EP claimed
EP-1422218-A1 ANTIVIRAL AGENT SHIONOGI & CO., LTD. (JP) 2004-05-26 EP claimed
WO-2003052106-A1 METHOD OF SCREENING COMPOUNDS CHILDREN'S MEDICAL CENTER CORPORATION (US) 2003-06-26 WO claimed
US-20030045479-A1 Novel N-formyl hydroxylamine compounds, compositions and methods of use VICURON HOLDINGS LLC 2003-03-06 US claimed
US-5939568-A Accelerated catalysis of olefinic epoxidations THE SCRIPPS RESEARCH INSTITUTE (US) 1999-08-17 US claimed
WO-1998033786-A9 ACCELERATED CATALYSIS OF OLEFINIC EPOXIDATIONS 1998-12-30 WO claimed
WO-1998033786-A1 ACCELERATED CATALYSIS OF OLEFINIC EPOXIDATIONS THE SCRIPPS RESEARCH INSTITUTE (US) 1998-08-06 WO claimed
US-4101507-A WITH PICOLINAMIDES AND ZINC OXIDE OR MAGNESIUM OXIDE THE FIRESTONE TIRE & RUBBER COMPANY (US) 1978-07-18 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10287255-B2 Compounds as histone deacetylase 6 inhibitors and pharmaceutical compositions comprising the same HDAC6, HDAC1, HDAC11 EGLN2 1706/4885FTO 4799/4885KDM4E 319/4885
US-20220008414-A1 PHARMACEUTICAL COMPOSITION COMPRISING HISTONE DEACETYLASE 6 INHIBITORS HDAC6, HDAC1, HDAC3 EGLN2 1159/4885FTO 4864/4885KDM4E 1264/4885
US-20030045479-A1 Novel N-formyl hydroxylamine compounds, compositions and methods of use PDF, HNMT, AADAC EGLN2 222/4885FTO 472/4885KDM4E 2350/4885
US-20110123434-A1 COMBINATION THERAPIES COMPRISING QUINOXALINE INHIBITORS OF P13K-ALPHA FOR USE IN THE TREATMENT OF CANCER TP53, PHKG1, TNNI3K EGLN2 1029/4885FTO 4750/4885KDM4E 835/4885
US-20160194321-A1 PYRROLOPYRIDINE OR PYRAZOLOPYRIDINE DERIVATIVES CHRM1, CHRM2, CHRM3 EGLN2 2435/4885FTO 881/4885KDM4E 2597/4885
US-20170096405-A1 NOVEL COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME HDAC6, HDAC1, HDAC5 EGLN2 3516/4885FTO 4806/4885KDM4E 468/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.