SCHEMBL3249440

SCHEMBL3249440

CCOC(=O)Oc1c[nH]c2c(=O)[nH]c3ccc(-c4cccc(NS(C)(=O)=O)c4)cc3c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.39
MMP13 P45452 1/20 0.39
POLB P06746 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ALDH1A1 P00352 2/20 0.38
LMNA P02545 2/20 0.38
TP53 P04637 1/20 0.38
GAA P10253 1/20 0.38
MAPK1 P28482 1/20 0.38
CYP1A2 P05177 3/20 0.38
CYP3A4 P08684 3/20 0.38
TDP2 O95551 2/20 0.38
CLK4 Q9HAZ1 2/20 0.38
USP2 O75604 1/20 0.38
TSHR P16473 1/20 0.38
HIF1A Q16665 1/20 0.38
BRD4 O60885 5/20 0.37
AAK1 Q2M2I8 1/20 0.37
DHFR P00374 1/20 0.37
ABL1 P00519 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3254540 0.90 MMP2 (0.46) MMP2MMP13POLBALDH1A1GAA
SCHEMBL3252205 0.89 TTK (0.42) MMP13SMN1; SMN2ALDH1A1HPGD
SCHEMBL3250925 0.87 NR1H2 (0.38) SMN1; SMN2ALDH1A1CYP1A2TSHRCYP2D6
SCHEMBL3251203 0.86 JAK3 (0.47) MMP2MMP13POLBJAK3
SCHEMBL3249063 0.86 CDK2 (0.39) LMNATSHRBRD4
SCHEMBL3252380 0.86 CSF1R (0.43) SMN1; SMN2ALDH1A1LMNAGAACYP1A2
SCHEMBL3252050 0.85 GAA (0.40) ALDH1A1LMNAGAAJAK3HPGD
SCHEMBL3243042 0.84 CYP17A1 (0.41) BRD4JAK3
SCHEMBL3249476 0.84 ICMT (0.37) SMN1; SMN2ALDH1A1LMNATP53GAA
SCHEMBL3243041 0.84 WEE1 (0.38) MMP2POLBALDH1A1LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899335-B1 PYRROLOQUINOLINE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS PF MEDICAMENT (FR) 2010-05-19 EP claimed