SCHEMBL3250449

SCHEMBL3250449

CN(C)C(=O)N(C(=O)OCc1ccccc1)c1ccc(-c2cn[nH]c2)cc1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 17/20 0.56
ROCK1 Q13464 3/20 0.44
MYLK4 Q86YV6 1/20 0.44
AKT1 P31749 1/20 0.41
AKT2 P31751 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
CYP2C9 P11712 1/20 0.40
CDC42BPA Q5VT25 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3249289 0.87 ROCK2 (0.61) ROCK2ROCK1CYP2C9CDC42BPA
SCHEMBL3250294 0.81 ROCK2 (0.54) ROCK2ROCK1MYLK4CYP2C9CDC42BPA
SCHEMBL3241309 0.79 ROCK2 (0.49) ROCK2ROCK1MYLK4CYP2C9CDC42BPA
SCHEMBL3239739 0.78 ROCK2 (0.53) ROCK2ROCK1MYLK4CYP2C9CDC42BPA
SCHEMBL3244750 0.78 ROCK2 (0.51) ROCK2ROCK1MYLK4CYP2C9CDC42BPA
SCHEMBL3248274 0.72 ROCK2 (1.00) ROCK2ROCK1MYLK4
SCHEMBL3252034 0.71 ROCK2 (0.48) ROCK2ROCK1MYLK4CYP2C9CDC42BPA
SCHEMBL3250445 0.70 ROCK2 (0.63) ROCK2ROCK1MYLK4
SCHEMBL9118903 0.70 ALDH1A1 (0.55) ALDH1A1MAPTHPGD
SCHEMBL3237795 0.70 ROCK2 (0.47) ROCK2ROCK1MYLK4CYP2C9CDC42BPA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010036316-A1 UREA AND CARBAMATE COMPOUNDS AND ANALOGS AS KINASE INHIBITORS FENG YANGBO (US) 2010-04-01 WO claimed