SCHEMBL3252241

SCHEMBL3252241

Oc1ncnc2nc(-c3ccccc3)cnc12

nearest known ligand 0.67

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PIK3CG P48736 4/20 0.48
ADK P55263 3/20 0.44
NOS1 P29475 1/20 0.42
BCHE P06276 1/20 0.40
MIF P14174 1/20 0.40
NPC1 O15118 1/20 0.39
PDGFRB P09619 1/20 0.39
KDR P35968 1/20 0.39
FLT3 P36888 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dimethylamine SCHEMBL11470117 0.94 PIK3CG (0.44) PIK3CGADKNOS1NPC1PDGFRB
SCHEMBL11472836 0.84 PIK3CG (0.47) PIK3CGADKNPC1RAB9ASMN1; SMN2
SCHEMBL11470380 0.84 ADK (0.56) PIK3CGADKNPC1RAB9ASMN1; SMN2
SCHEMBL11478905 0.82 PIK3CG (0.48) PIK3CGADK
SCHEMBL11467366 0.82 BCHE (0.53) PIK3CGADKBCHE
SCHEMBL11470116 0.80 ADK (0.71) PIK3CGADKNOS1
SCHEMBL11446163 0.80 ADK (0.67) PIK3CGADKNOS1
SCHEMBL11467784 0.76 ALDH1A1 (0.47) ADKNOS1NPC1RAB9ASMN1; SMN2
SCHEMBL4361291 0.76 PIK3CG (0.53) PIK3CGADKNOS1SMN1; SMN2
SCHEMBL13019092 0.72 CSF1R (0.54) ADKRAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1511852-B1 USE OF FLUORINE NMR FOR HIGH THROUGHPUT SCREENING NERVIANO MEDICAL SCIENCES SRL (IT) 2010-05-26 EP disclosed
US-7470543-B2 Methods for identifying ligands using competitive binding 1H NMR experiments NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2008-12-30 US disclosed
EP-1511852-A4 USE OF FLUORINE NMR FOR HIGH THROUGHPUT SCREENING PHARMACIA & UPJOHN CO LLC (US) 2008-07-16 EP disclosed
CN-1668757-A Use of fluorine nmr for high throughput screening UPJOHN CO (US) 2005-09-14 CN disclosed
EP-1511988-A4 METHODS FOR IDENTIFYING LIGANDS USING COMPETITIVE BINDING sp 1 /sp H NMR EXPERIMENTS PHARMACIA & UPJOHN CO LLC (US) 2005-07-06 EP disclosed
EP-1511988-A1 METHODS FOR IDENTIFYING LIGANDS USING COMPETITIVE BINDING sp 1 /sp H NMR EXPERIMENTS PHARMACIA & UPJOHN COMPANY (US) 2005-03-09 EP disclosed
EP-1511852-A2 USE OF FLUORINE NMR FOR HIGH THROUGHPUT SCREENING PHARMACIA & UPJOHN COMPANY (US) 2005-03-09 EP disclosed
WO-2004051214-A2 USE OF FLUORINE NMR FOR HIGH THROUGHPUT SCREENING PHARMACIA & UPJOHN COMPANY (US) 2004-06-17 WO disclosed
US-20040091937-A1 Use of fluorine NMR for high throughput screening NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2004-05-13 US disclosed
US-20040072362-A1 Methods for identifying ligands using competitive binding 1H NMR experiments PHARMACIA & UPJOHN COMPANY 2004-04-15 US disclosed
WO-2003104778-A1 METHODS FOR IDENTIFYING LIGANDS USING COMPETITIVE BINDING 1H NMR EXPERIMENTS PHARMACIA & UPJOHN COMPANY (US) 2003-12-18 WO disclosed
US-4183934-A NONALIURETIC DIURETICS ABBOTT LABORATORIES (US) 1980-01-15 US disclosed