SCHEMBL3253786

SCHEMBL3253786

O=C(OC1(Cc2ccccc2Br)NC(c2ccccc2)C(c2ccccc2)N1)C(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.33
ALDH1A1 P00352 1/20 0.33
RAB9A P51151 1/20 0.33
HCRTR2 O43614 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
P2RX7 Q99572 1/20 0.31
TP53 P04637 1/20 0.31
MMP1 P03956 1/20 0.30
MMP2 P08253 1/20 0.30
MMP9 P14780 1/20 0.30
MMP12 P39900 1/20 0.30
FFAR1 O14842 1/20 0.30
FFAR4 Q5NUL3 1/20 0.30
HDAC4 P56524 1/20 0.30
KDM1A O60341 1/20 0.30
PTGDR2 Q9Y5Y4 1/20 0.30
SIGMAR1 Q99720 1/20 0.30
PPARG P37231 1/20 0.30
PPARA Q07869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3255401 0.87 P2RX7 (0.39) GAAALDH1A1RAB9AMEN1KMT2A
SCHEMBL3255382 0.86 CYP1A2 (0.37) GAAALDH1A1RAB9AMEN1KMT2A
SCHEMBL3256042 0.86 P2RX7 (0.39) GAAALDH1A1RAB9AP2RX7FFAR1
SCHEMBL3256647 0.84 P2RX7 (0.34) GAARAB9AP2RX7TP53FFAR4
SCHEMBL3258301 0.81 GAA (0.38) GAAALDH1A1RAB9AMEN1KMT2A
SCHEMBL3256107 0.81 KMT2A (0.39) ALDH1A1RAB9AMEN1KMT2ATP53
SCHEMBL3254057 0.81 TP53 (0.42) GAARAB9AMEN1KMT2AP2RX7
SCHEMBL3254884 0.81 SIGMAR1 (0.35) GAAALDH1A1TP53SIGMAR1PPARG
SCHEMBL3255278 0.81 SIGMAR1 (0.35) GAAMEN1KMT2AP2RX7TP53
SCHEMBL3258687 0.80 GPBAR1 (0.39) GAAKMT2AKDM1ASIGMAR1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651613-B1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS AVENTIS PHARMA INC (US) 2010-05-26 EP disclosed