SCHEMBL3256647

SCHEMBL3256647

O=C(OC1(Cc2cccc(F)c2F)NC(c2ccccc2)C(c2ccccc2)N1)C(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.34
GRIN2B Q13224 1/20 0.32
GAA P10253 2/20 0.32
RIPK1 Q13546 1/20 0.32
CTSL P07711 1/20 0.32
ELANE P08246 1/20 0.32
CTSG P08311 1/20 0.32
CTSS P25774 1/20 0.32
FFAR4 Q5NUL3 1/20 0.31
ALKBH1 Q13686 1/20 0.31
CXCL8 P10145 1/20 0.30
PTGS2 P35354 1/20 0.30
PDE10A Q9Y233 1/20 0.30
TP53 P04637 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3255401 0.92 P2RX7 (0.39) P2RX7GAACTSLELANECTSG
SCHEMBL3256725 0.87 GAA (0.33) P2RX7GAATP53RAB9A
SCHEMBL3255413 0.84 ALDH1A1 (0.38) P2RX7TP53RAB9A
SCHEMBL3255382 0.84 CYP1A2 (0.37) P2RX7GAARAB9A
SCHEMBL3253786 0.84 GAA (0.33) P2RX7GAAFFAR4TP53RAB9A
SCHEMBL3256042 0.84 P2RX7 (0.39) P2RX7GAARAB9A
SCHEMBL3255278 0.83 SIGMAR1 (0.35) P2RX7GAARIPK1TP53
SCHEMBL3254884 0.83 SIGMAR1 (0.35) GRIN2BGAARIPK1TP53
SCHEMBL3248922 0.83 P2RX7 (0.38) P2RX7GAACTSLELANECTSG
SCHEMBL3254166 0.82 SMN1; SMN2 (0.39) GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651613-B1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS AVENTIS PHARMA INC (US) 2010-05-26 EP disclosed