SCHEMBL3255382

SCHEMBL3255382

O=C(OC1(Cc2ccccc2Cl)NC(c2ccccc2)C(c2ccccc2)N1)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C9 P11712 2/20 0.37
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
CYP2C19 P33261 2/20 0.37
SLC6A3 Q01959 2/20 0.37
HSD11B1 P28845 1/20 0.37
P2RX7 Q99572 1/20 0.35
GAA P10253 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
ALDH1A1 P00352 2/20 0.34
HPGD P15428 1/20 0.34
KCNJ5 P48544 2/20 0.33
KCNJ3 P48549 2/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3258306 0.88 P2RX7 (0.39) CYP1A2CYP3A4CYP2D6CYP2C9SLC6A2
SCHEMBL3255755 0.88 ALDH1A1 (0.36) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL3255401 0.87 P2RX7 (0.39) P2RX7GAARAB9AALDH1A1KCNH2
SCHEMBL3256042 0.86 P2RX7 (0.39) P2RX7GAARAB9AALDH1A1HPGD
SCHEMBL3253786 0.86 GAA (0.33) P2RX7GAARAB9AALDH1A1MEN1
SCHEMBL3255018 0.84 GAA (0.35) GAARAB9AALDH1A1MEN1KMT2A
SCHEMBL3254166 0.84 SMN1; SMN2 (0.39) GAAALDH1A1MEN1KMT2A
SCHEMBL3256647 0.84 P2RX7 (0.34) P2RX7GAARAB9A
SCHEMBL3256757 0.82 RPA1 (0.34) GAANPC1RAB9AMAPK1
SCHEMBL3256107 0.81 KMT2A (0.39) NPC1RAB9AALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651613-B1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS AVENTIS PHARMA INC (US) 2010-05-26 EP disclosed