SCHEMBL3255405

SCHEMBL3255405

COc1ccc(CCC2(OC(=O)C(F)(F)F)NC(c3ccccc3)C(c3ccccc3)N2)cc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
RAB9A P51151 2/20 0.40
NPC1 O15118 1/20 0.40
GAA P10253 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ATM Q13315 1/20 0.39
FABP7 O15540 1/20 0.38
FABP5 Q01469 1/20 0.38
EDNRA P25101 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALOX15 P16050 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
GPR52 Q9Y2T5 1/20 0.38
FPR2 P25090 1/20 0.38
ALOX5 P09917 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3258744 0.89 P2RX7 (0.38) ALDH1A1MEN1KMT2AFABP7FABP5
SCHEMBL3253969 0.89 CYP2C19 (0.41) ALDH1A1GAAMEN1KMT2AKDM4E
SCHEMBL3258633 0.88 PDPK1 (0.41) KMT2AATMKDM4E
SCHEMBL3255825 0.88 PDPK1 (0.36) ALDH1A1GAAMEN1KMT2A
SCHEMBL3253833 0.84 CES1 (0.41) RAB9AKDM4E
SCHEMBL3254386 0.83 CES1 (0.43) RAB9AKDM4E
SCHEMBL3258350 0.83 SLC6A2 (0.39) RAB9ANPC1MEN1KMT2AATM
SCHEMBL3258561 0.83 PDPK1 (0.39) MEN1KMT2AATMTDP1
SCHEMBL3257098 0.82 TAAR1 (0.39) KMT2A
SCHEMBL3248922 0.82 P2RX7 (0.38) ALDH1A1GAAMEN1KMT2AALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651613-B1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS AVENTIS PHARMA INC (US) 2010-05-26 EP disclosed