SCHEMBL3258561

SCHEMBL3258561

O=C(OC1(CCc2ccc(Cl)c(Cl)c2)NC(c2ccccc2)C(c2ccccc2)N1)C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.39
PLAAT3 P53816 1/20 0.35
PLAAT5 Q96KN8 1/20 0.35
PLAAT2 Q9NWW9 1/20 0.35
PLAAT4 Q9UL19 1/20 0.35
TRPV1 Q8NER1 2/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
RECQL P46063 1/20 0.35
BLM P54132 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CHRM5 P08912 2/20 0.34
CHRM1 P11229 2/20 0.34
CHRM3 P20309 2/20 0.34
TSHR P16473 1/20 0.34
TBXA2R P21731 1/20 0.34
PTGER1 P34995 1/20 0.34
PTGER4 P35408 1/20 0.34
PTGFR P43088 1/20 0.34
PTGER3 P43115 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3251176 0.90 ALDH1A1 (0.35) PDPK1TRPV1TSHRSIGMAR1
SCHEMBL3255825 0.88 PDPK1 (0.36) PDPK1MEN1KMT2A
SCHEMBL3258394 0.87 P2RX7 (0.42) PLAAT3PLAAT5PLAAT2PLAAT4TRPV1
SCHEMBL3258744 0.84 P2RX7 (0.38) PLAAT3PLAAT5PLAAT2PLAAT4MEN1
SCHEMBL3253810 0.84 ALDH1A1 (0.41) PLAAT3PLAAT5PLAAT2PLAAT4MEN1
SCHEMBL3256757 0.84 RPA1 (0.34)
SCHEMBL3259233 0.84 P2RX7 (0.41) CHRM3CHRM2
SCHEMBL3258306 0.84 P2RX7 (0.39) PLAAT3PLAAT5PLAAT2PLAAT4TRPV1
SCHEMBL3258633 0.84 PDPK1 (0.41) PDPK1PLAAT3PLAAT5PLAAT2PLAAT4
SCHEMBL3258350 0.83 SLC6A2 (0.39) MEN1KMT2ACHRM3CHRM2ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651613-B1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS AVENTIS PHARMA INC (US) 2010-05-26 EP disclosed