SCHEMBL3248922

SCHEMBL3248922

O=C(OC1(CCc2ccccc2F)NC(c2ccccc2)C(c2ccccc2)N1)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.38
TRPV1 Q8NER1 1/20 0.35
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
TAAR1 Q96RJ0 3/20 0.34
LMNA P02545 1/20 0.34
CTSL P07711 1/20 0.34
ELANE P08246 1/20 0.34
CTSG P08311 1/20 0.34
CTSS P25774 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
SCN3A Q9NY46 5/20 0.32
KCNH2 Q12809 4/20 0.32
SCN1A P35498 1/20 0.32
SCN4A P35499 1/20 0.32
SCN7A Q01118 1/20 0.32
SCN5A Q14524 1/20 0.32
SCN9A Q15858 1/20 0.32
SCN2A Q99250 1/20 0.32
SCN8A Q9UQD0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3251110 0.90 ALDH1A1 (0.37) TRPV1TAAR1LMNAL3MBTL1ALDH1A1
SCHEMBL3255401 0.88 P2RX7 (0.39) P2RX7TRPV1KMT2AMEN1CTSL
SCHEMBL3258306 0.87 P2RX7 (0.39) P2RX7TRPV1KCNH2GAAALDH1A1
SCHEMBL3257098 0.86 TAAR1 (0.39) KMT2ATAAR1
SCHEMBL3258744 0.84 P2RX7 (0.38) P2RX7KMT2AMEN1LMNAALDH1A1
SCHEMBL3256647 0.83 P2RX7 (0.34) P2RX7CTSLELANECTSGCTSS
SCHEMBL3255405 0.82 ALDH1A1 (0.41) KMT2AMEN1GAAALDH1A1ALOX5
SCHEMBL3256725 0.81 GAA (0.33) P2RX7LMNAGAASMN1; SMN2
SCHEMBL3253833 0.81 CES1 (0.41) P2RX7LMNAL3MBTL1SMN1; SMN2
SCHEMBL3259233 0.81 P2RX7 (0.41) P2RX7TAAR1LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651613-B1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS AVENTIS PHARMA INC (US) 2010-05-26 EP disclosed