SCHEMBL3258744

SCHEMBL3258744

O=C(OC1(CCc2ccc(F)cc2)NC(c2ccccc2)C(c2ccccc2)N1)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.38
TP53 P04637 1/20 0.36
FABP7 O15540 1/20 0.36
FABP5 Q01469 1/20 0.36
KDM1A O60341 1/20 0.35
RCOR1 Q9UKL0 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.33
PLAAT3 P53816 1/20 0.33
PLAAT5 Q96KN8 1/20 0.33
PLAAT2 Q9NWW9 1/20 0.33
PLAAT4 Q9UL19 1/20 0.33
LTA4H P09960 1/20 0.33
EPHX2 P34913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3248358 0.90 ALDH1A1 (0.38) P2RX7ALDH1A1LMNA
SCHEMBL3255825 0.90 PDPK1 (0.36) TP53KDM1ARCOR1ALDH1A1KMT2A
SCHEMBL3258633 0.90 PDPK1 (0.41) KDM1AKDM4EKMT2APLAAT3PLAAT5
SCHEMBL3254057 0.89 TP53 (0.42) P2RX7TP53FABP7FABP5KDM1A
SCHEMBL3255405 0.89 ALDH1A1 (0.41) FABP7FABP5KDM4EALDH1A1KMT2A
SCHEMBL3259233 0.88 P2RX7 (0.41) P2RX7ALDH1A1LMNA
SCHEMBL3253833 0.86 CES1 (0.41) P2RX7SLC6A3KDM4ELMNAEPHX2
SCHEMBL3254386 0.85 CES1 (0.43) P2RX7SLC6A3KDM4ELMNAEPHX2
SCHEMBL3258561 0.84 PDPK1 (0.39) KMT2AMEN1PLAAT3PLAAT5PLAAT2
SCHEMBL3248922 0.84 P2RX7 (0.38) P2RX7ALDH1A1KMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1651613-B1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS AVENTIS PHARMA INC (US) 2010-05-26 EP disclosed