SCHEMBL3257301

SCHEMBL3257301

O=C(O)CC(CC1CCN(C(=O)c2cccc([AsH]C3=NCCN3)c2)CC1)c1cccc(F)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 5/20 0.49
ITGAV P06756 5/20 0.49
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 1/20 0.38
TDP1 Q9NUW8 1/20 0.37
HSD11B1 P28845 1/20 0.36
ITGA2B P08514 2/20 0.36
USP2 O75604 3/20 0.36
CYP3A4 P08684 2/20 0.36
TSHR P16473 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
EGLN1 Q9GZT9 1/20 0.35
HTT P42858 1/20 0.35
MGLL Q99685 1/20 0.35
GAA P10253 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2925480 0.83 ITGB3 (0.50) ITGB3ITGAVALDH1A1KDM4ETDP1
SCHEMBL2925340 0.75 ITGB3 (0.42) ITGB3ITGAVALDH1A1ITGA2BMGLL
SCHEMBL547914 0.66 ITGB3 (1.00) ITGB3ITGAVITGA2B
SCHEMBL2906666 0.66 ITGB3 (1.00) ITGB3ITGAVITGA2B
SCHEMBL2917750 0.65 ITGB3 (0.91) ITGB3ITGAVITGA2B
SCHEMBL5857867 0.62 GABBR2 (0.50) ITGB3ITGAV
SCHEMBL4919120 0.61 SIGMAR1 (0.49) ALDH1A1KDM4ETDP1HSD11B1USP2
SCHEMBL10154308 0.60 ITGB3 (0.41) ITGB3ITGAV
SCHEMBL2503391 0.60 OPRK1 (0.44) ITGB3ITGAVKDM4E
SCHEMBL1244906 0.60 SMN1; SMN2 (0.69) ALDH1A1KDM4ETDP1HSD11B1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2217569-A1 ENANTIOSELECTIVE PROCESS FOR PREPARING A SUBSTITUTED ALKANOIC ACID Janssen Pharmaceutica N.V. (BE) 2010-08-18 EP disclosed
WO-2009058314-A1 ENANTIOSELECTIVE PROCESS FOR PREPARING A SUBSTITUTED ALKANOIC ACID JANSSEN PHARMACEUTICA, N.V. (BE) 2009-05-07 WO disclosed