SCHEMBL3258696

SCHEMBL3258696

CCOC(=O)C1(N[C@H](C)c2ccccc2)CCC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.49
CYP3A4 P08684 2/20 0.46
CYP2C19 P33261 2/20 0.46
LMNA P02545 1/20 0.44
HPGD P15428 1/20 0.44
KCNA3 P22001 1/20 0.44
OPRM1 P35372 5/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP2C9 P11712 1/20 0.43
TSHR P16473 1/20 0.43
RECQL P46063 1/20 0.43
MMP8 P22894 1/20 0.43
OPRD1 P41143 3/20 0.42
OPRK1 P41145 3/20 0.42
SLC22A1 O15245 1/20 0.42
SLC6A4 P31645 1/20 0.42
ADRA1A P35348 1/20 0.42
KCNH2 Q12809 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3258693 1.00 SMN1; SMN2 (0.49) SMN1; SMN2CYP3A4CYP2C19LMNAHPGD
SCHEMBL13483586 0.82 MME (0.50) SMN1; SMN2CYP3A4CYP2C19LMNAHPGD
SCHEMBL3259891 0.81 LMNA (0.51) LMNAHPGDALDH1A1RECQLMEN1
SCHEMBL3259889 0.81 LMNA (0.51) LMNAHPGDALDH1A1RECQLMEN1
SCHEMBL14960649 0.79 SMN1; SMN2 (0.40) SMN1; SMN2CYP3A4CYP2C19LMNAOPRM1
SCHEMBL11155829 0.76 CYP3A4 (0.42) SMN1; SMN2CYP3A4CYP2C19KCNA3OPRM1
SCHEMBL15461468 0.76 ALDH1A1 (0.37) SMN1; SMN2CYP3A4CYP2C19LMNAOPRM1
SCHEMBL15461485 0.75 ALDH1A1 (0.36) SMN1; SMN2CYP3A4CYP2C19OPRM1ALDH1A1
SCHEMBL15461439 0.74 ALDH1A1 (0.38) SMN1; SMN2CYP3A4CYP2C19LMNAOPRM1
SCHEMBL2083186 0.74 APAF1 (0.43) SMN1; SMN2CYP3A4CYP2C19KCNA3OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE41149-E1 Stereoisomerically pure 7-[(7S)-7-amino-5-azaspiro[2.4]heptan-5-yl]-6-fluoro-1-[(1R,2S)-2-fluoro-1-cyclopropyl]-8-methoxy-1,4-dihydro-4-oxo-3-quinolinecarboxylic acid or a pharmaceutically acceptable salt thereof; antibacterial agents DAIICHI SANKYO COMPANY, LIMITED (JP) 2010-02-23 US disclosed
US-6031102-A Optically active pyridonecarboxylic acid derivatives DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2000-02-29 US disclosed
US-5587386-A BACTERICIDES, MICROBIOCIDES DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1996-12-24 US disclosed