SCHEMBL3260672

SCHEMBL3260672

O=C(CC1CN(C(=O)O)CCN1)OC1CCCNc2ccccc21

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
REN P00797 3/20 0.35
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA4 P22748 2/20 0.34
CA9 Q16790 2/20 0.34
PARP1 P09874 1/20 0.33
CXCR4 P61073 4/20 0.33
F12 P00748 5/20 0.32
F2 P00734 2/20 0.32
CACNA2D1 P54289 1/20 0.31
CACNA1B Q00975 1/20 0.31
CACNB1 Q02641 1/20 0.31
ADRB1 P08588 1/20 0.31
HSD11B1 P28845 1/20 0.31
OPRM1 P35372 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3264285 0.79 LTA4H (0.33)
SCHEMBL7835340 0.72 ALDH1A1 (0.33) F12F2
SCHEMBL28639323 0.68 F12 (0.36) F12F2
SCHEMBL900236 0.68 REN (0.42) RENCA1CA2CA4CA9
SCHEMBL20141289 0.68 REN (0.42) RENCA1CA2CA4CA9
SCHEMBL10565873 0.67 F12 (0.40) F12F2
SCHEMBL5719329 0.67 CA1 (0.62) RENCA1CA2CA4CA9
SCHEMBL4749948 0.67 CA1 (0.62) RENCA1CA2CA4CA9
SCHEMBL3495230 0.67 CA1 (0.62) RENCA1CA2CA4CA9
SCHEMBL4288512 0.66 LTA4H (0.52) RENCA1CA2CA4CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170831-A1 BENZAZEPINE DERIVATIVES USEFUL AS VASOPRESSIN ANTAGONISTS Otsuka Pharmaceutical Co., Ltd. (JP) 2010-04-07 EP disclosed
WO-2009001968-A1 BENZAZEPINE DERIVATIVES USEFUL AS VASOPRESSIN ANTAGONISTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-12-31 WO disclosed