SCHEMBL3261071

SCHEMBL3261071

CCCN[C@@H](CC(N)=O)C(N)=O

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ECE1 P42892 4/20 0.40
ALOX15 P16050 1/20 0.33
MMP1 P03956 1/20 0.33
MMP2 P08253 1/20 0.33
MMP3 P08254 1/20 0.33
MMP9 P14780 1/20 0.33
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CTSD P07339 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3261068 1.00 ECE1 (0.40) ECE1ALOX15MMP1MMP2MMP3
SCHEMBL29697562 0.88 ALOX15 (0.44) ECE1ALOX15MMP2CA1CA2
SCHEMBL7355950 0.86 NOD1 (0.40) ECE1ALOX15CA1CA2
SCHEMBL30089038 0.86 ECE1 (0.44) ECE1ALOX15CA1CA2
SCHEMBL8728335 0.86 GPR84 (0.33) ECE1ALOX15MMP1MMP2MMP3
SCHEMBL23831532 0.85 EPHX1 (0.42) ALOX15
SCHEMBL1045359 0.85 EPHX1 (0.42) ALOX15
SCHEMBL1045358 0.85 EPHX1 (0.42) ALOX15
SCHEMBL29364715 0.85 EPHX1 (0.42) ALOX15
SCHEMBL2692730 0.85 EPHX1 (0.42) ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2106279-A2 STATIONARY PHASE GRADIENT CHROMATOGRAPHY Cryobiophysica, Inc. (US) 2009-10-07 EP claimed
US-20080179243-A1 Stationary Phase Gradient Chromatography HIRSH ALLEN 2008-07-31 US claimed
WO-2008086357-A2 STATIONARY PHASE GRADIENT CHROMATOGRAPHY CRYOBIOPHYSICA, INC. (US) 2008-07-17 WO claimed
US-20250084181-A1 PERTUZUMAB VARIANTS AND EVALUATION THEREOF GENENTECH, INC. (US) 2025-03-13 US disclosed
WO-2024105205-A1 ANTIBODY-DRUG CONJUGATES (A2DCS) WITH ENZYMATICALLY CLEAVABLE GROUPS BAYER AKTIENGESELLSCHAFT (DE) 2024-05-23 WO disclosed
US-20100151501-A1 Forms of Prostate Specific Antigens and Methods for their Detection HYBRITECH INCORPORATED 2010-06-17 US disclosed
US-7659073-B2 Forms of prostate specific antigens and methods for their detection HYBRITECH INCORPORATED (US) 2010-02-09 US disclosed
EP-2106279-A2 STATIONARY PHASE GRADIENT CHROMATOGRAPHY Cryobiophysica, Inc. (US) 2009-10-07 EP disclosed
EP-1392719-B1 FORMS OF PROSTATE SPECIFIC ANTIGENS AND METHODS FOR THEIR DETECTION HYBRITECH INC (US) 2009-04-22 EP disclosed
EP-0981629-B1 FORMS OF PROSTATE SPECIFIC ANTIGEN AND METHODS FOR THEIR DETECTION HYBRITECH INC (US) 2008-08-13 EP disclosed
US-20080179243-A1 Stationary Phase Gradient Chromatography HIRSH ALLEN 2008-07-31 US disclosed
US-20020058291-A1 Forms of prostate specific antigens and methods for their detection HYBRITECH INCORPORATED 2002-05-16 US disclosed
US-20020045198-A1 Forms of prostate specific antigens and methods for their detection HYBRITECH INCORPORATED 2002-04-18 US disclosed
EP-1175619-A1 METHOD TO DISTINGUISH PROSTATE CANCER FROM BENIGN PROSTATIC HYPERPLASIA Hybritech Incorporated (US) 2002-01-30 EP disclosed
EP-1173556-A1 FORMS OF PROSTATE SPECIFIC ANTIGEN (PSA) SPECIFIC FOR BENIGN PROSTATIC HYPERPLASIA (BPH) AND METHODS OF USING SUCH Hybritech Incorporated (US) 2002-01-23 EP disclosed
WO-2000066718-A1 FORMS OF PROSTATE SPECIFIC ANTIGEN (PSA) SPECIFIC FOR BENIGN PROSTATIC HYPERPLASIA (BPH) AND METHODS OF USING SUCH HYBRITECH INCORPORATED (US) 2000-11-09 WO disclosed
WO-2000067030-A1 METHOD TO DISTINGUISH PROSTATE CANCER FROM BENIGN PROSTATIC HYPERPLASIA HYBRITECH INCORPORATED (US) 2000-11-09 WO disclosed
EP-0981629-A1 FORMS OF PROSTATE SPECIFIC ANTIGEN AND METHODS FOR THEIR DETECTION HYBRITECH INCORPORATED (US) 2000-03-01 EP disclosed
WO-1998049323-A1 FORMS OF PROSTATE SPECIFIC ANTIGEN AND METHODS FOR THEIR DETECTION HYBRITECH INCORPORATED (US) 1998-11-05 WO disclosed
US-5260060-A Dissolving blood clots, anticoagulant, metalloproteinase UNIVERSITY OF SOUTHERN CALIFORNIA (US) 1993-11-09 US disclosed