SCHEMBL3261864

SCHEMBL3261864

O=c1[nH][nH]cc1-c1ccc(Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.46
GAA P10253 3/20 0.42
ALDH1A1 P00352 2/20 0.42
MAPT P10636 1/20 0.42
THRB P10828 1/20 0.42
TSHR P16473 1/20 0.42
NPC1 O15118 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
MAP4K4 O95819 2/20 0.40
PTGS2 P35354 2/20 0.39
PTGS1 P23219 1/20 0.39
MCL1 Q07820 1/20 0.39
LMNA P02545 1/20 0.38
RAB9A P51151 1/20 0.38
KIF11 P52732 1/20 0.37
GSK3B P49841 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
AHR P35869 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3263382 0.78 ALDH1A1 (0.53) KDM4EGAAALDH1A1MAPTTHRB
SCHEMBL4872103 0.73 GAA (0.60) KDM4EGAAALDH1A1MAPTTHRB
SCHEMBL28409089 0.73 MEN1 (0.48) KDM4EGAAALDH1A1MAPTNPC1
SCHEMBL29809206 0.72 ALDH1A1 (0.67) KDM4EGAAALDH1A1MAPTTSHR
SCHEMBL3262685 0.69 GSK3B (0.51) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL3561082 0.69 MAPT (0.48) KDM4EGAAALDH1A1MAPTTHRB
SCHEMBL11685438 0.66 MCL1 (0.45) KDM4EGAAALDH1A1MAPTTHRB
SCHEMBL11689636 0.65 ALDH1A1 (0.47) KDM4EGAAALDH1A1MAPTNPC1
SCHEMBL11308251 0.64
Sulfuric Acid SCHEMBL11767295 0.64 CYP1A2 (0.52) ALDH1A1MEN1KMT2APTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010015656-A2 NEW ALKOXYPYRAZOLES INSTITUT PASTEUR (FR) 2010-02-11 WO disclosed
WO-2010015656-A2 NEW ALKOXYPYRAZOLES INSTITUT PASTEUR (FR) 2010-02-11 WO disclosed
EP-2151434-A1 Alkoxypyrazoles and the process for their preparation Institut Pasteur (FR) 2010-02-10 EP disclosed