SCHEMBL3262463

SCHEMBL3262463

NC(=O)C(Oc1ccccc1F)c1cccnc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.44
ALDH1A1 P00352 2/20 0.42
GAA P10253 1/20 0.42
POLB P06746 1/20 0.41
SLC6A2 P23975 2/20 0.40
SLC6A4 P31645 2/20 0.40
SLC6A3 Q01959 2/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PPARG P37231 2/20 0.39
PPARA Q07869 2/20 0.39
LMNA P02545 1/20 0.39
CFTR P13569 1/20 0.38
GOPC Q9HD26 1/20 0.38
PARP10 Q53GL7 1/20 0.38
TSHR P16473 1/20 0.38
SGMS2 Q8NHU3 1/20 0.37
F7 P08709 1/20 0.37
F3 P13726 1/20 0.37
SARM1 Q6SZW1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17968476 0.84 PPARG (0.52) ALDH1A1GAASLC6A2SLC6A4SLC6A3
SCHEMBL28741054 0.74 HTT (0.46) NOTUMALDH1A1SLC6A2SLC6A4SLC6A3
SCHEMBL19716861 0.74 LMNA (0.46) ALDH1A1POLBSLC6A2SLC6A4SLC6A3
SCHEMBL4496453 0.72 PLA2G7 (0.43) ALDH1A1POLBSLC6A2SLC6A4SLC6A3
SCHEMBL5660114 0.72 ALDH1A1 (0.44) ALDH1A1GAASLC6A2SLC6A4SLC6A3
SCHEMBL21881179 0.71 PPARA (0.68) ALDH1A1GAASLC6A2SLC6A4SLC6A3
SCHEMBL306372 0.70 F7 (0.53) ALDH1A1GAAPOLBSLC6A2SLC6A4
SCHEMBL28341455 0.70 ALDH1A1 (0.53) ALDH1A1GAAHTTSMN1; SMN2PPARG
SCHEMBL362393 0.69 F7 (0.52) ALDH1A1GAASLC6A2SLC6A4SLC6A3
SCHEMBL29937752 0.68 ALDH1A1 (0.55) ALDH1A1SLC6A2SLC6A4SLC6A3HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010015387-A1 DAA-PYRIDINE AS PERIPHERAL BENZODIAZEPINE RECEPTOR LIGAND FOR DIAGNOSTIC IMAGING AND PHARMACEUTICAL TREATMENT BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-02-11 WO disclosed
WO-2010015340-A1 DAA-PYRIDINE AS PERIPHERAL BENZODIAZEPINE RECEPTOR LIGAND FOR DIAGNOSTIC IMAGING AND PHARMACEUTICAL TREATMENT BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-02-11 WO disclosed