SCHEMBL3265091

SCHEMBL3265091

CCC(C)C(NC(=O)c1nc(-c2ccc(N)cc2)no1)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.47
GAA P10253 1/20 0.47
CA2 P00918 3/20 0.46
CA1 P00915 2/20 0.46
HDAC4 P56524 2/20 0.41
AKR1B1 P15121 1/20 0.41
POLB P06746 1/20 0.40
SMPD1 P17405 1/20 0.40
SCN10A Q9Y5Y9 1/20 0.40
TP53 P04637 3/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
RXFP1 Q9HBX9 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
ACACB O00763 1/20 0.39
PPARD Q03181 1/20 0.39
PPARA Q07869 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3265775 0.85 LMNA (0.45) KDM4EGAACA2CA1HDAC4
SCHEMBL3265444 0.84 CSGALNACT1 (0.54) SMN1; SMN2LMNAMAPT
SCHEMBL2297789 0.81 KDM4E (0.47) KDM4EGAAHDAC4SMPD1SCN10A
SCHEMBL3266079 0.77 CSGALNACT1 (0.60) SMN1; SMN2LMNAMAPT
SCHEMBL2296375 0.74 CSGALNACT1 (0.65)
SCHEMBL2296367 0.74 CSGALNACT1 (0.65)
SCHEMBL1756198 0.73 MASP2 (0.44) KDM4ECA2CA1AKR1B1TP53
SCHEMBL3265094 0.73 KDM4E (0.52) KDM4EGAAHDAC4POLBSMPD1
SCHEMBL2299081 0.72 DGAT1 (0.56)
SCHEMBL2299944 0.71 CSGALNACT1 (0.66)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010023609-A1 OXAZOLE, OXADIAZOLE AND THIAZOLE DERIVATIVES AS DIACYLGLYCEROL ACYLTRANFERASE INHIBITORS PIRAMAL LIFE SCIENCES LIMITED (IN) 2010-03-04 WO disclosed