SCHEMBL3265646

SCHEMBL3265646

Cn1ncn(-c2ccccc2)c1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 2/20 0.45
GSK3B P49841 2/20 0.45
NFE2L2 Q16236 1/20 0.44
MAPT P10636 1/20 0.41
ALDH1A1 P00352 5/20 0.40
CYP1A2 P05177 2/20 0.40
KDM4E B2RXH2 1/20 0.40
HPGD P15428 1/20 0.40
BLM P54132 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
PGR P06401 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
PPARG P37231 1/20 0.39
PPARD Q03181 1/20 0.39
PPARA Q07869 1/20 0.39
HCAR1 Q9BXC0 1/20 0.39
MITF O75030 1/20 0.39
LMNA P02545 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7471419 0.82 NFE2L2 (0.45) GSK3AGSK3BNFE2L2MAPTALDH1A1
SCHEMBL22349810 0.81 MAPT (0.64) GSK3AGSK3BMAPTALDH1A1HPGD
SCHEMBL16197227 0.81 NPC1 (0.44) GSK3AGSK3BMAPTALDH1A1KDM4E
SCHEMBL20644484 0.78 ALDH1A1 (0.48) MAPTALDH1A1KDM4EHPGDTDP1
SCHEMBL14280089 0.78 MAPT (0.51) GSK3AGSK3BMAPTALDH1A1CYP1A2
SCHEMBL7477352 0.77 MAPT (0.39) MAPTALDH1A1KDM4ESMN1; SMN2PPARG
SCHEMBL22931495 0.76 HTT (0.41) GSK3AGSK3BMAPTALDH1A1CYP1A2
SCHEMBL22349850 0.76 ALDH1A1 (0.47) GSK3AGSK3BALDH1A1TDP1SMN1; SMN2
SCHEMBL14600370 0.76 ROCK2 (0.50) GSK3AGSK3BMAPTALDH1A1CYP1A2
SCHEMBL22931489 0.74 KDM4E (0.44) NFE2L2ALDH1A1KDM4ETDP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010025870-A1 SYNERGISTIC COMBINATIONS OF THIADIAZOL CARBONIC ACID DERIVATIVES BAYER CROPSCIENCE AG (DE) 2010-03-11 WO claimed
US-7166603-B2 Dihydropyrimidone inhibitors of calcium channel function BRISTOL-MYERS SQUIBB CO. (US) 2007-01-23 US disclosed
WO-2005009392-A2 DIHYDROPYRIMIDONE INHIBITORS OF CALCIUM CHANNEL FUNCTION BRISTOL-MYERS SQUIBB COMPANY (US) 2005-02-03 WO disclosed